Therapeutic discovery for marrow failure with MDS predisposition using pluripotent stem cells

JCI Insight. 2019 Apr 30;5(12):e125157. doi: 10.1172/jci.insight.125157.

Abstract

Monosomy 7 or deletion of 7q (del(7q)) are common clonal cytogenetic abnormalities associated with high grade myelodysplastic syndrome (MDS) arising in inherited and acquired bone marrow failure. Current non-transplant approaches to treat marrow failure may be complicated by stimulation of clonal outgrowth. To study the biological consequences of del(7q) within the context of a failing marrow, we generated induced pluripotent stem cells (iPSCs) derived from patients with Shwachman Diamond Syndrome (SDS), a bone marrow failure disorder with MDS predisposition, and genomically engineered a 7q deletion. The TGFβ pathway was the top differentially regulated pathway in transcriptomic analysis of SDS versus SDSdel(7q) iPSCs. SMAD2 phosphorylation was increased in SDS relative to wild type cells consistent with hyperactivation of the TGFbeta pathway in SDS. Phospho-SMAD2 levels were reduced following 7q deletion in SDS cells and increased upon restoration of 7q diploidy. Inhibition of the TGFbeta pathway rescued hematopoiesis in SDS-iPSCs and in bone marrow hematopoietic cells from SDS patients while it had no impact on the SDSdel(7q) cells. These results identified a potential targetable vulnerability to improve hematopoiesis in an MDS-predisposition syndrome, and highlight the importance of the germline context of somatic alterations to inform precision medicine approaches to therapy.

Keywords: Bone marrow; Drug therapy; Hematology; Human stem cells; Therapeutics.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, Non-P.H.S.

MeSH terms

  • Bone Marrow / drug effects
  • Bone Marrow / pathology*
  • Cell Engineering
  • Chromosome Deletion
  • Chromosomes, Human, Pair 7 / genetics
  • HEK293 Cells
  • Hematopoiesis / drug effects
  • Hematopoiesis / genetics
  • Hematopoietic Stem Cells / drug effects
  • Hematopoietic Stem Cells / pathology
  • Humans
  • Induced Pluripotent Stem Cells / drug effects
  • Induced Pluripotent Stem Cells / pathology
  • Karyotyping
  • Myelodysplastic Syndromes / genetics
  • Myelodysplastic Syndromes / prevention & control*
  • Phosphorylation / genetics
  • Precision Medicine / methods*
  • RNA-Seq
  • Shwachman-Diamond Syndrome / diagnosis
  • Shwachman-Diamond Syndrome / genetics
  • Shwachman-Diamond Syndrome / pathology
  • Shwachman-Diamond Syndrome / therapy*
  • Signal Transduction / drug effects
  • Signal Transduction / genetics
  • Smad2 Protein / metabolism
  • Transforming Growth Factor beta / metabolism

Substances

  • SMAD2 protein, human
  • Smad2 Protein
  • Transforming Growth Factor beta

Supplementary concepts

  • Chromosome 7, monosomy