Identification of a USP9X Substrate NFX1-123 by SILAC-Based Quantitative Proteomics

J Proteome Res. 2019 Jun 7;18(6):2654-2665. doi: 10.1021/acs.jproteome.9b00139. Epub 2019 May 22.

Abstract

The deubiquitinase USP9X is involved in multiple diseases including neurodegeneration, epilepsy, and various types of tumors by targeting different substrates. In the present study, we aimed to explore the potential substrates of USP9X and performed SILAC-based quantitative proteomics to compare these substrates in USP9X-knockdown and wild-type HeLa cells. We consequently carried out Flag-NFX1-123 tag affinity-based mass spectrometry and confirmed that the X-box binding nuclear factor NFX1-123 interacted with USP9X. Moreover, immunoprecipitation assays verified a direct interaction between USP9X and NFX1-123. Further experiments confirmed that NFX1-123 could be modified by ubiquitination and that USP9X stabilized NFX1-123 via efficient deubiquitination of NFX1-123. Knockdown of USP9X resulted in decreased NFX1-123 protein levels compared with their unchanged corresponding mRNA levels in different cell lines. In summary, we found that NFX1-123 was a bona fide substrate of the deubiquitinase USP9X and that it could be degraded by the ubiquitin-proteasome system. The present study provided new insight into understanding the biological function of USP9X by targeting its substrate NFX1-123.

Keywords: NFX1-123; SILAC; USP9X; deubiquitinase; quantitative proteomics.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Apoptosis / genetics
  • Cell Proliferation / genetics
  • Gene Expression Regulation / genetics
  • Gene Knockdown Techniques
  • HeLa Cells
  • Humans
  • Nerve Degeneration / genetics*
  • Nerve Degeneration / pathology
  • Proteasome Endopeptidase Complex / genetics
  • Proteasome Endopeptidase Complex / metabolism
  • Proteomics*
  • Repressor Proteins / genetics*
  • Ubiquitin / genetics
  • Ubiquitin Thiolesterase / genetics*
  • Ubiquitination / genetics

Substances

  • NFX1 protein, human
  • Repressor Proteins
  • USP9X protein, human
  • Ubiquitin
  • Ubiquitin Thiolesterase
  • Proteasome Endopeptidase Complex