Dimethyl fumarate therapy reduces memory T cells and the CNS migration potential in patients with multiple sclerosis

Mult Scler Relat Disord. 2020 Jan:37:101451. doi: 10.1016/j.msard.2019.101451. Epub 2019 Oct 16.

Abstract

Background: Dimethyl fumarate (DMF) is a disease-modifying therapy for patients with relapsing-remitting multiple sclerosis (RRMS). T cells are major contributors to the pathogenesis of RRMS, where they regulate the pathogenic immune response and participate in CNS lesion development.

Objectives: In this study we evaluate the therapeutic effects of DMF on T cell subpopulations, their CNS migration potential and effector functions.

Methods: Blood and CSF from untreated and DMF-treated patients with RRMS and healthy donors were analyzed by flow cytometry.

Results: DMF reduced the prevalence of circulating proinflammatory CD4+ and CD8+ memory T cells, whereas regulatory T cells were unaffected. Furthermore, DMF reduced the frequency of CD4+ T cells expressing CNS-homing markers. In coherence, we found a reduced recruitment of CD4+ but not CD8+ T cells to CSF. We also found that monomethyl fumarate dampened T cell proliferation and reduced the frequency of TNF-α, IL-17 and IFN-γ producing T cells.

Conclusion: DMF influences the balance between proinflammatory and regulatory T cells, presumably favoring a less proinflammatory environment. DMF also reduces the CNS migratory potential of CD4+ T cells whereas CD8+ T cells are less affected. Altogether, our study suggests an anti-inflammatory effect of DMF mainly on the CD4+ T cell compartment.

MeSH terms

  • Adult
  • Cell Proliferation / drug effects
  • Cohort Studies
  • Cytokines / drug effects*
  • Dimethyl Fumarate / pharmacology*
  • Female
  • Fumarates / pharmacology*
  • Humans
  • Immunologic Factors / pharmacology*
  • Inflammation / blood
  • Inflammation / cerebrospinal fluid
  • Inflammation / drug therapy*
  • Inflammation / immunology
  • Male
  • Middle Aged
  • Multiple Sclerosis, Relapsing-Remitting / blood
  • Multiple Sclerosis, Relapsing-Remitting / cerebrospinal fluid
  • Multiple Sclerosis, Relapsing-Remitting / drug therapy*
  • Multiple Sclerosis, Relapsing-Remitting / immunology
  • T-Lymphocytes / drug effects*
  • Young Adult

Substances

  • Cytokines
  • Fumarates
  • Immunologic Factors
  • monomethyl fumarate
  • Dimethyl Fumarate