Engaging chromatin: PRC2 structure meets function

Br J Cancer. 2020 Feb;122(3):315-328. doi: 10.1038/s41416-019-0615-2. Epub 2019 Nov 11.

Abstract

Polycomb repressive complex 2 (PRC2) is a key epigenetic multiprotein complex involved in the regulation of gene expression in metazoans. PRC2 is formed by a tetrameric core that endows the complex with histone methyltransferase activity, allowing it to mono-, di- and tri-methylate histone H3 on lysine 27 (H3K27me1/2/3); H3K27me3 is a hallmark of facultative heterochromatin. The core complex of PRC2 is bound by several associated factors that are responsible for modulating its targeting specificity and enzymatic activity. Depletion and/or mutation of the subunits of this complex can result in severe developmental defects, or even lethality. Furthermore, mutations of these proteins in somatic cells can be drivers of tumorigenesis, by altering the transcriptional regulation of key tumour suppressors or oncogenes. In this review, we present the latest results from structural studies that have characterised PRC2 composition and function. We compare this information with data and literature for both gain-of function and loss-of-function missense mutations in cancers to provide an overview of the impact of these mutations on PRC2 activity.

Publication types

  • Research Support, Non-U.S. Gov't
  • Review

MeSH terms

  • Animals
  • Chromatin / metabolism*
  • Enhancer of Zeste Homolog 2 Protein / genetics
  • Enhancer of Zeste Homolog 2 Protein / metabolism
  • Enhancer of Zeste Homolog 2 Protein / ultrastructure
  • Gain of Function Mutation
  • Gene Expression Regulation, Neoplastic / genetics*
  • Histone Code / genetics*
  • Humans
  • Loss of Function Mutation
  • Mice
  • Neoplasm Proteins
  • Neoplasms / genetics*
  • Polycomb Repressive Complex 2 / genetics*
  • Polycomb Repressive Complex 2 / metabolism
  • Polycomb Repressive Complex 2 / ultrastructure
  • Protein Domains
  • Protein Structure, Quaternary
  • Protein Structure, Tertiary
  • Protein Subunits
  • Structure-Activity Relationship
  • Transcription Factors

Substances

  • Chromatin
  • EED protein, human
  • Eed protein, mouse
  • Neoplasm Proteins
  • Protein Subunits
  • SUZ12 protein, human
  • Suz12 protein, mouse
  • Transcription Factors
  • EZH1 protein, human
  • Enhancer of Zeste Homolog 2 Protein
  • Ezh1 protein, mouse
  • Polycomb Repressive Complex 2