In Silico Discovery and Validation of Neuropeptide-Y-Binding Peptides for Sensors

J Phys Chem B. 2020 Jan 9;124(1):61-68. doi: 10.1021/acs.jpcb.9b09439. Epub 2019 Dec 26.

Abstract

Wearable sensors for human health, performance, and state monitoring, which have a linear response to the binding of biomarkers found in sweat, saliva, or urine, are of current interest for many applications. A critical part of any device is a biological recognition element (BRE) that is able to bind a biomarker at the surface of a sensor with a high affinity and selectivity to produce a measurable signal response. In this study, we discover and compare 12-mer peptides that bind to neuropeptide Y (NPY), a stress and human health biomarker, using independent and complimentary experimental and computational approaches. The affinities of the NPY-binding peptides discovered by both methods are equivalent and below the micromolar level, which makes them suitable for application in sensors. The in silico design protocol for peptide-based BREs is low cost, highly efficient, and simple, suggesting its utility for discovering peptide binders to a variety of biomarker targets.

Publication types

  • Research Support, U.S. Gov't, Non-P.H.S.

MeSH terms

  • Algorithms
  • Amino Acid Sequence
  • Biomarkers / metabolism
  • Humans
  • Kinetics
  • Molecular Dynamics Simulation
  • Neuropeptide Y / analysis
  • Neuropeptide Y / chemistry
  • Neuropeptide Y / metabolism*
  • Peptides / chemistry
  • Peptides / metabolism*
  • Protein Binding
  • Protein Structure, Secondary

Substances

  • Biomarkers
  • Neuropeptide Y
  • Peptides