TRIB3 supports breast cancer stemness by suppressing FOXO1 degradation and enhancing SOX2 transcription

Nat Commun. 2019 Dec 16;10(1):5720. doi: 10.1038/s41467-019-13700-6.

Abstract

The existence of breast cancer stem cells (BCSCs) is a major reason underlying cancer metastasis and recurrence after chemotherapy and radiotherapy. Targeting BCSCs may ameliorate breast cancer relapse and therapy resistance. Here we report that expression of the pseudokinase Tribble 3 (TRIB3) positively associates with breast cancer stemness and progression. Elevated TRIB3 expression supports BCSCs by interacting with AKT to interfere with the FOXO1-AKT interaction and suppress FOXO1 phosphorylation, ubiquitination, and degradation by E3 ligases SKP2 and NEDD4L. The accumulated FOXO1 promotes transcriptional expression of SOX2, a transcriptional factor for cancer stemness, which in turn, activates FOXO1 transcription and forms a positive regulatory loop. Disturbing the TRIB3-AKT interaction suppresses BCSCs by accelerating FOXO1 degradation and reducing SOX2 expression in mouse models of breast cancer. Our study provides insights into breast cancer development and confers a potential therapeutic strategy against TRIB3-overexpressed breast cancer.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Breast / pathology
  • Breast Neoplasms / genetics*
  • Breast Neoplasms / pathology
  • Cell Cycle Proteins / metabolism*
  • Cell Line, Tumor
  • Disease Progression
  • Female
  • Forkhead Box Protein O1 / metabolism*
  • Gene Expression Regulation, Neoplastic
  • Humans
  • Mice
  • Middle Aged
  • Neoplastic Stem Cells / pathology*
  • Protein Binding
  • Protein Serine-Threonine Kinases / antagonists & inhibitors*
  • Protein Serine-Threonine Kinases / metabolism
  • Proteolysis
  • Proto-Oncogene Proteins c-akt / metabolism
  • Repressor Proteins / metabolism*
  • SOXB1 Transcription Factors / genetics*
  • Tissue Array Analysis
  • Transcription, Genetic
  • Xenograft Model Antitumor Assays

Substances

  • Cell Cycle Proteins
  • FOXO1 protein, human
  • Forkhead Box Protein O1
  • Repressor Proteins
  • SOX2 protein, human
  • SOXB1 Transcription Factors
  • TRIB3 protein, human
  • Protein Serine-Threonine Kinases
  • Proto-Oncogene Proteins c-akt