Omega-3 fatty acids as regulators of brown/beige adipose tissue: from mechanisms to therapeutic potential

J Physiol Biochem. 2020 May;76(2):251-267. doi: 10.1007/s13105-019-00720-5. Epub 2019 Dec 18.

Abstract

Adipose tissue dysfunction represents the hallmark of obesity. Brown/beige adipose tissues play a crucial role in maintaining energy homeostasis through non-shivering thermogenesis. Brown adipose tissue (BAT) activity has been inversely related to body fatness, suggesting that BAT activation is protective against obesity. BAT plays also a key role in the control of triglyceride clearance, glucose homeostasis, and insulin sensitivity. Therefore, BAT/beige activation has been proposed as a strategy to prevent or ameliorate obesity development and associated commorbidities. In the last few years, a variety of preclinical studies have proposed n-3 polyunsaturated fatty acids (n-3 PUFAs) as novel inducers of BAT activity and white adipose tissue browning. Here, we review the in vitro and in vivo available evidences of the thermogenic properties of n-3 PUFAs, especially focusing on the molecular and cellular physiological mechanisms involved. Finally, we also discuss the challenges and future perspectives to better characterize the therapeutic potential of n-3 PUFAs as browning agents, especially in humans.

Keywords: Adipose tissue; Browning; Obesity; n-3 PUFAs.

Publication types

  • Review

MeSH terms

  • Adipose Tissue, Beige / metabolism*
  • Adipose Tissue, Brown / metabolism*
  • Animals
  • Cells, Cultured
  • Energy Metabolism
  • Fatty Acids, Omega-3* / pharmacology
  • Fatty Acids, Omega-3* / physiology
  • Humans
  • Mice
  • Obesity* / drug therapy
  • Obesity* / metabolism
  • Rats
  • Thermogenesis

Substances

  • Fatty Acids, Omega-3