Inhibition of Dectin-1 in mice ameliorates cardiac remodeling by suppressing NF-κB/NLRP3 signaling after myocardial infarction

Int Immunopharmacol. 2020 Mar:80:106116. doi: 10.1016/j.intimp.2019.106116. Epub 2020 Jan 21.

Abstract

The myocardial inflammatory response is a consequence of myocardial infarction (MI), which may deteriorate cardiac remodeling and lead to dysfunction in the heart post-MI. Dectin-1 is a c-type lectin, which has been shown to regulate innate immune responses to pathogens. However, the role of Dectin-1 in the heart diseases remains largely unknown. In this study, we aimed to investigate the effects of Dectin-1 on cardiac remodeling post-MI. We found that cardiac Dectin-1 mRNA and protein expressions were significantly elevated in C57BL/6 mice after MI. In vitro, hypoxia induced cardiomyocyte injury in parallel with increased Dectin-1 protein expression. Knockdown of Dectin-1 remarkably attenuated cardiomyocyte death under hypoxia and lipopolysaccharide (LPS) stimulation. In vivo administration of adeno-associated virus serotype 9 mediated silencing of Dectin-1, which significantly decreased cardiac fibrosis, dilatation, and improved cardiac function in the mice post-MI. At the molecular level, downregulation of Dectin-1 dramatically suppressed up-regulation of nuclear factor-κB (NF-κB), nucleotide-binding oligomerization domain-like receptor family pyrin domain-containing 3 (NLRP3), and the inflammatory genes involved in fibrogenesis and cardiac remodeling after MI. Furthermore, treatment with BAY11-7082, an inhibitor of NF-κB, repressed the activation of NF-κB, and attenuated LPS induced elevation of NLRP3 and cell death in cardiomyocytes. Collectively, upregulation of Dectin-1 in cardiomyocytes post-MI contributes to cardiac remodeling and cardiac dysfunction at least partially by activating NF-κB and NLRP3. This study identified Dectin-1 as a promising therapeutic target for ischemic heart disease.

Keywords: Dectin-1; Inflammation; Myocardial infarction; NF-κB; NLRP3.

MeSH terms

  • Animals
  • Disease Models, Animal
  • Down-Regulation
  • Female
  • Gene Knockdown Techniques
  • Humans
  • Lectins, C-Type / genetics
  • Lectins, C-Type / metabolism*
  • Lipopolysaccharides / immunology
  • Male
  • Mice
  • Myocardial Infarction / drug therapy
  • Myocardial Infarction / immunology*
  • Myocardial Infarction / pathology
  • Myocardium / cytology
  • Myocardium / immunology
  • Myocardium / pathology
  • Myocytes, Cardiac
  • NF-kappa B / antagonists & inhibitors
  • NF-kappa B / metabolism
  • NLR Family, Pyrin Domain-Containing 3 Protein / metabolism
  • Nitriles / pharmacology
  • Nitriles / therapeutic use
  • Primary Cell Culture
  • RNA, Small Interfering / metabolism
  • Signal Transduction / drug effects
  • Signal Transduction / genetics
  • Signal Transduction / immunology*
  • Sulfones / pharmacology
  • Sulfones / therapeutic use
  • Up-Regulation / immunology
  • Ventricular Remodeling / drug effects
  • Ventricular Remodeling / genetics
  • Ventricular Remodeling / immunology*

Substances

  • 3-(4-methylphenylsulfonyl)-2-propenenitrile
  • Lectins, C-Type
  • Lipopolysaccharides
  • NF-kappa B
  • NLR Family, Pyrin Domain-Containing 3 Protein
  • Nitriles
  • Nlrp3 protein, mouse
  • RNA, Small Interfering
  • Sulfones
  • dectin 1