Three new diterpenoids from Euphorbia peplus

Nat Prod Res. 2021 Nov;35(21):3901-3907. doi: 10.1080/14786419.2020.1749609. Epub 2020 Apr 14.

Abstract

Three new diterpenoids (1-3) (two abietane type diterpenoids and a paralianone type diterpenoid), together with four known compounds (4-7) were isolated from the whole plants of Euphorbia peplus. Their structures were elucidated through spectroscopic analysis and physicochemical characteristics. The cytotoxic activities of compounds 1-7 against five human tumour cell lines were evaluated, however, they were inactive at the concentration of 40 μM. The compound 3 enhanced lysosomal biogenesis with Lyso Tracker staining intensity of 132.6%.

Keywords: Euphorbia peplus; Euphorbiaceae; ent-abietane diterpenoids; paralianone diterpenoids.

MeSH terms

  • Abietanes
  • Antineoplastic Agents, Phytogenic* / pharmacology
  • Diterpenes* / pharmacology
  • Euphorbia*
  • Humans
  • Molecular Structure

Substances

  • Abietanes
  • Antineoplastic Agents, Phytogenic
  • Diterpenes