QT interval prolongation related to afatinib treatment in a patient with metastatic non-small-cell lung cancer

Curr Probl Cancer. 2020 Dec;44(6):100594. doi: 10.1016/j.currproblcancer.2020.100594. Epub 2020 May 27.

Abstract

Afatinib improves survival in metastatic non-small-cell lung cancer driven by activating epidermal growth factor receptor mutations. QT interval prolongation is a possible side effect of targeted anticancer drugs, but this has not been reported before with afatinib. We report a case of metastatic pulmonary adenocarcinoma with epidermal growth factor receptor exon 19 deletion who was treated with first-line afatinib. The patient was started on afatinib with a total dose of 40 mg/day and experienced grade 3 (>500 ms) QT interval prolongation in the seventh week. Dose was interrupted and then reduced to 30 mg/day after the event repeated. QT prolongation occurred only once with the reduced dose and radiologic oligoprogression was detected. Local therapy was performed and afatinib was continued as 30 mg/day. To the best of our knowledge, this case marks the first QT interval prolongation associated with afatinib. It is prudent to perform a baseline cardiologic evaluation and electrocardiogram monitoring in non-small cell lung cancer patients treated with this drug.

Keywords: Afatinib; Epidermal growth factor receptor; Non–small-cell lung cancer; QT prolongation; Tyrosine kinase inhibitor.

Publication types

  • Case Reports

MeSH terms

  • Adult
  • Afatinib / adverse effects*
  • Antineoplastic Agents / adverse effects*
  • Carcinoma, Non-Small-Cell Lung / drug therapy*
  • Carcinoma, Non-Small-Cell Lung / pathology
  • Female
  • Humans
  • Long QT Syndrome / chemically induced
  • Long QT Syndrome / pathology*
  • Lung Neoplasms / drug therapy*
  • Lung Neoplasms / pathology
  • Prognosis

Substances

  • Antineoplastic Agents
  • Afatinib