A general method to optimize and functionalize red-shifted rhodamine dyes

Nat Methods. 2020 Aug;17(8):815-821. doi: 10.1038/s41592-020-0909-6. Epub 2020 Jul 27.

Abstract

Expanding the palette of fluorescent dyes is vital to push the frontier of biological imaging. Although rhodamine dyes remain the premier type of small-molecule fluorophore owing to their bioavailability and brightness, variants excited with far-red or near-infrared light suffer from poor performance due to their propensity to adopt a lipophilic, nonfluorescent form. We report a framework for rationalizing rhodamine behavior in biological environments and a general chemical modification for rhodamines that optimizes long-wavelength variants and enables facile functionalization with different chemical groups. This strategy yields red-shifted 'Janelia Fluor' (JF) dyes useful for biological imaging experiments in cells and in vivo.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Cell Line, Tumor
  • Fluorescent Dyes / chemistry*
  • Humans
  • Infrared Rays
  • Microscopy, Fluorescence / methods
  • Molecular Structure
  • Rhodamines / chemistry*

Substances

  • Fluorescent Dyes
  • Rhodamines