Evaluation of a TrkB agonist on spatial and motor learning in the Ube3a mouse model of Angelman syndrome

Learn Mem. 2020 Aug 17;27(9):346-354. doi: 10.1101/lm.051201.119. Print 2020 Sep.

Abstract

Angelman syndrome is a rare neurodevelopmental disorder caused by a mutation in the maternal allele of the gene Ube3a The primary symptoms of Angelman syndrome are severe cognitive deficits, impaired motor functions, and speech disabilities. Analogous phenotypes have been detected in young adult Ube3a mice. Here, we investigate cognitive phenotypes of Ube3a mice as compared to wild-type littermate controls at an older adult age. Water maze spatial learning, swim speed, and rotarod motor coordination and balance were impaired at 6 mo of age, as predicted. Based on previous findings of reduced brain-derived neurotrophic factor in Ube3a mice, a novel therapeutic target, the TrkB agonist 7,8-DHF, was interrogated. Semichronic daily treatment with 7,8-DHF, 5 mg/kg i.p., did not significantly improve the impairments in performance during the acquisition of the water maze hidden platform location in Ube3a mice, after training with either massed or spaced trials, and had no effect on the swim speed and rotarod deficits. Robust behavioral phenotypes in middle-aged Ube3a mice appear to result from continued motor decline. Our results suggest that motor deficits could offer useful outcome measures for preclinical testing of many pharmacological targets, with the goal of reducing symptoms in adults with Angelman syndrome.

Publication types

  • Evaluation Study
  • Research Support, N.I.H., Extramural

MeSH terms

  • Age Factors
  • Angelman Syndrome / drug therapy*
  • Animals
  • Behavior, Animal / drug effects*
  • Disease Models, Animal
  • Female
  • Flavones / pharmacology*
  • Male
  • Maze Learning / drug effects*
  • Membrane Glycoproteins / agonists*
  • Mice
  • Mice, Knockout
  • Motor Activity / drug effects*
  • Phenotype
  • Protein-Tyrosine Kinases
  • Ubiquitin-Protein Ligases

Substances

  • 6,7-dihydroxyflavone
  • Flavones
  • Membrane Glycoproteins
  • Ube3a protein, mouse
  • Ubiquitin-Protein Ligases
  • Ntrk2 protein, mouse
  • Protein-Tyrosine Kinases