A broad-spectrum virus- and host-targeting peptide against respiratory viruses including influenza virus and SARS-CoV-2

Nat Commun. 2020 Aug 25;11(1):4252. doi: 10.1038/s41467-020-17986-9.

Abstract

The 2019 novel respiratory virus (SARS-CoV-2) causes COVID-19 with rapid global socioeconomic disruptions and disease burden to healthcare. The COVID-19 and previous emerging virus outbreaks highlight the urgent need for broad-spectrum antivirals. Here, we show that a defensin-like peptide P9R exhibited potent antiviral activity against pH-dependent viruses that require endosomal acidification for virus infection, including the enveloped pandemic A(H1N1)pdm09 virus, avian influenza A(H7N9) virus, coronaviruses (SARS-CoV-2, MERS-CoV and SARS-CoV), and the non-enveloped rhinovirus. P9R can significantly protect mice from lethal challenge by A(H1N1)pdm09 virus and shows low possibility to cause drug-resistant virus. Mechanistic studies indicate that the antiviral activity of P9R depends on the direct binding to viruses and the inhibition of virus-host endosomal acidification, which provides a proof of concept that virus-binding alkaline peptides can broadly inhibit pH-dependent viruses. These results suggest that the dual-functional virus- and host-targeting P9R can be a promising candidate for combating pH-dependent respiratory viruses.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Amino Acid Sequence
  • Animals
  • Antiviral Agents / chemistry
  • Antiviral Agents / metabolism
  • Antiviral Agents / pharmacology*
  • Antiviral Agents / therapeutic use
  • Cell Line
  • Coronavirus / drug effects*
  • Endosomes / chemistry
  • Endosomes / drug effects
  • Female
  • Humans
  • Hydrogen-Ion Concentration
  • Influenza A virus / drug effects*
  • Influenza A virus / metabolism
  • Mice
  • Mice, Inbred BALB C
  • Orthomyxoviridae Infections / drug therapy
  • Orthomyxoviridae Infections / metabolism
  • Peptides / chemistry
  • Peptides / metabolism
  • Peptides / pharmacology*
  • Peptides / therapeutic use
  • Protein Binding
  • Protein Conformation
  • Rhinovirus / drug effects
  • Rhinovirus / metabolism
  • Viral Load / drug effects
  • Virus Replication / drug effects

Substances

  • Antiviral Agents
  • Peptides