SCF FBXW17 E3 ubiquitin ligase regulates FBXL19 stability and cell migration

J Cell Biochem. 2021 Apr;122(3-4):326-334. doi: 10.1002/jcb.29860. Epub 2020 Oct 14.

Abstract

The Skp1-Cul1-F-box protein (SCF) E3 ligase complex is one of the largest ubiquitin E3 ligase families. FBXL19, a F-box protein in SCFFBXL19 E3 ligase complex, regulates a variety of cellular responses including cell migration. We have shown that FBXL19 is not stable and its degradation is mediated by the ubiquitin-proteasome system, while the ubiquitin E3 ligase for FBXL19 ubiquitination and degradation has not been identified. In the study, we discovered that a new ubiquitin E3 ligase, SCFFBXW17 , ubiquitinates and induces FBXL19 degradation. Exogenous FBXW17 targets FBXL19 for its ubiquitination and degradation. Lysine 114 in FBXL19 is a potential ubiquitin acceptor site. Acetylation of FBXL19 attenuated SCFFBXW17 -mediated FBXL19 degradation. SCFFBXL19 E3 ligase reduced Rac1 levels and cell migration, while the effects were attenuated by exogenous FBXW17. Downregulation of FBXW17 attenuated lysophosphatidic acid-induced lamellipodia formation and Rac1 accumulation at migration leading edge. Taken together with our previous studies, FBXL19 is degraded by the ubiquitin-proteasome system and its site-specific ubiquitination is mediated by SCFFBXW17 E3 ligase, which promotes cell migration.

Keywords: F-box protein; SCF E3 ligase; cell migration; protein degradation; ubiquitination.

Publication types

  • Research Support, N.I.H., Extramural

MeSH terms

  • Acetylation
  • Animals
  • Cell Line
  • Cell Movement / genetics
  • Cell Movement / physiology*
  • DNA-Binding Proteins / genetics
  • DNA-Binding Proteins / metabolism*
  • F-Box Proteins / genetics
  • F-Box Proteins / metabolism*
  • Immunoblotting
  • Immunoprecipitation
  • Mice
  • RNA, Small Interfering / genetics
  • RNA, Small Interfering / metabolism
  • Ubiquitination / genetics
  • Ubiquitination / physiology
  • rac1 GTP-Binding Protein / genetics
  • rac1 GTP-Binding Protein / metabolism

Substances

  • DNA-Binding Proteins
  • F-Box Proteins
  • FBXL19 protein, mouse
  • RNA, Small Interfering
  • rac1 GTP-Binding Protein