Cortical projection neurons as a therapeutic target in multiple sclerosis

Expert Opin Ther Targets. 2020 Dec;24(12):1211-1224. doi: 10.1080/14728222.2020.1842358. Epub 2020 Nov 8.

Abstract

Introduction: Multiple sclerosis (MS) is a chronic inflammatory-demyelinating disease of the central nervous system associated with lesions of the cortical gray matter and subcortical white matter. Recently, cortical lesions have become a major focus of research because cortical pathology and neuronal damage are critical determinants of irreversible clinical progression. Recent transcriptomic studies point toward cell type-specific changes in cortical neurons in MS with a selective vulnerability of excitatory projection neuron subtypes.

Areas covered: We discuss the cortical mapping and the molecular properties of excitatory projection neurons and their role in MS lesion pathology while placing an emphasis on their subtype-specific transcriptomic changes and levels of vulnerability. We also examine the latest magnetic resonance imaging techniques to study cortical MS pathology as a key tool for monitoring disease progression and treatment efficacy. Finally, we consider possible therapeutic avenues and novel strategies to protect excitatory cortical projection neurons. Literature search methodology: PubMed articles from 2000-2020.

Expert opinion: Excitatory cortical projection neurons are an emerging therapeutic target in the treatment of progressive MS. Understanding neuron subtype-specific molecular pathologies and their exact spatial mapping will help establish starting points for the development of novel cell type-specific therapies and biomarkers in MS.

Keywords: Cortical projection neurons; cortical pathology; magnetic resonance imaging; multiple sclerosis; single-cell RNA-sequencing; transcriptomics.

Publication types

  • Research Support, Non-U.S. Gov't
  • Review

MeSH terms

  • Animals
  • Biomarkers / metabolism
  • Disease Progression
  • Humans
  • Magnetic Resonance Imaging
  • Molecular Targeted Therapy*
  • Multiple Sclerosis / diagnostic imaging
  • Multiple Sclerosis / physiopathology
  • Multiple Sclerosis / therapy*
  • Neurons / pathology*

Substances

  • Biomarkers