An analysis of genetic targets for guiding clinical management of follicular lymphoma

Expert Rev Hematol. 2020 Dec;13(12):1361-1372. doi: 10.1080/17474086.2020.1850252. Epub 2020 Dec 4.

Abstract

Introduction: Follicular lymphoma (FL) is one of the most common non-Hodgkin lymphoma (NHL) types, where genomic studies have accumulated potentially useful information about frequently mutated genes and deregulated pathways, which has allowed to a better understanding of the molecular pathogenesis of this tumor and the complex interrelationship between the tumoral cells and the stroma. Areas covered: The results of the molecular studies performed on Follicular Lymphoma have been here reviewed, summarizing the results of the clinical trials so far developed on this basis and discussing the reasons for the successes and failures. Searches were performed on June 1st, 2020, in PubMed and ClinicalTrials.gov. Expert opinion: Targeted therapy for follicular lymphoma has multiple opportunities including the use of epigenetic drugs, PI3K inhibitors, modifiers of the immune stroma and others. Data currently known on FL pathogenesis suggest that combining these treatments with immunotherapy should be explored in clinical trials, mainly for patients with clinical progression or adverse prognostic markers. Association of targeted trials with dynamic molecular studies of the tumor and serum samples is advised. Chemotherapy-free approaches should also be explored as first-line therapy for FL patients.

Keywords: BCL2 inhibitors; BCL6 inhibitors; epigenetic therapy; follicular lymphoma; targeted therapy.

Publication types

  • Research Support, Non-U.S. Gov't
  • Review

MeSH terms

  • Antineoplastic Combined Chemotherapy Protocols / therapeutic use*
  • B-Lymphocytes / pathology
  • Clinical Trials as Topic
  • Germinal Center / cytology
  • Humans
  • Immune Checkpoint Inhibitors / therapeutic use
  • Immunologic Factors / therapeutic use
  • Immunophenotyping
  • Immunotherapy, Adoptive
  • Lymphoma, Follicular / diagnosis
  • Lymphoma, Follicular / drug therapy*
  • Lymphoma, Follicular / genetics
  • Lymphoma, Follicular / pathology
  • Molecular Targeted Therapy*
  • Neoplasm Proteins / antagonists & inhibitors*
  • Neoplasm Proteins / genetics
  • Neoplasm Staging
  • Neoplastic Stem Cells / pathology
  • Prognosis
  • Protein Kinase Inhibitors / therapeutic use
  • Translocation, Genetic

Substances

  • Immune Checkpoint Inhibitors
  • Immunologic Factors
  • Neoplasm Proteins
  • Protein Kinase Inhibitors