Endogenous antisense RNA curbs CD39 expression in Crohn's disease

Nat Commun. 2020 Nov 18;11(1):5894. doi: 10.1038/s41467-020-19692-y.

Abstract

CD39 is an ectonucleotidase that initiates conversion of extracellular nucleotides into immunosuppressive adenosine. CD39 is expressed by regulatory T (Treg)-cells, where it mediates immunosuppression, and by a subset of T-helper (Th) 17-cells, where it limits pathogenicity. CD39 is regulated via single-nucleotide-polymorphisms and upon activation of aryl-hydrocarbon-receptor and oxygen-mediated pathways. Here we report a mechanism of CD39 regulation that relies on the presence of an endogenous antisense RNA, transcribed from the 3'-end of the human CD39/ENTPD1 gene. CD39-specific antisense is increased in Treg and Th17-cells of Crohn's disease patients over controls. It largely localizes in the cell nucleus and regulates CD39 by interacting with nucleolin and heterogeneous-nuclear-ribonucleoprotein-A1. Antisense silencing results in CD39 upregulation in vitro and amelioration of disease activity in a trinitro-benzene-sulfonic-acid model of colitis in humanized NOD/scid/gamma mice. Inhibition/blockade of antisense might represent a therapeutic strategy to restore CD39 along with immunohomeostasis in Crohn's disease.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, Non-P.H.S.

MeSH terms

  • Animals
  • Antigens, CD / genetics*
  • Antigens, CD / immunology
  • Apyrase / genetics*
  • Apyrase / immunology
  • Crohn Disease / genetics*
  • Crohn Disease / immunology
  • Female
  • Humans
  • Mice
  • Mice, Inbred NOD
  • RNA, Antisense / genetics*
  • RNA, Antisense / immunology
  • T-Lymphocytes, Regulatory / immunology
  • Th17 Cells / immunology

Substances

  • Antigens, CD
  • RNA, Antisense
  • Apyrase
  • CD39 antigen