The Cytotoxic Effect of α-Synuclein Aggregates

Chemphyschem. 2021 Mar 17;22(6):526-532. doi: 10.1002/cphc.202000831. Epub 2021 Feb 16.

Abstract

Parkinson's disease is a neurodegenerative disorder involving a functional protein, α-synuclein, whose primary function is related to vesicle trafficking. However, α-synuclein is prone to form aggregates, and these inclusions, known as Lewy bodies, are the hallmark of Parkinson's disease. α-synuclein can alter its conformation and acquire aggregating capacity, forming aggregates containing β-sheets. This protein's pathogenic importance is based on its ability to form oligomers that impair synaptic transmission and neuronal function by increasing membrane permeability and altering homeostasis, generating a deleterious effect over cells. First, we establish that oligomers interfere with the mechanical properties of 1,2-dioleoyl-sn-glycero-3-phosphocholine (DOPC) membrane, as demonstrated by nanoindentation curves. In contrast, nanoindentation revealed that the α-synuclein monomer's presence leads to a much more resistant lipid bilayer. Moreover, the oligomers' interaction with cell membranes can promote lactate dehydrogenase (LDH) release, suggesting the activation of cytotoxic events.

Keywords: Parkinson's disease; aggregates; membrane; nanoindentation; toxicity.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Cell Line, Tumor
  • Cell Membrane / drug effects*
  • Hydrophobic and Hydrophilic Interactions
  • L-Lactate Dehydrogenase / metabolism
  • Lipid Bilayers / chemistry
  • Lipid Bilayers / metabolism*
  • Mice
  • Phosphatidylcholines / chemistry
  • Protein Aggregates*
  • Protein Multimerization
  • alpha-Synuclein / chemistry
  • alpha-Synuclein / metabolism*
  • alpha-Synuclein / toxicity*

Substances

  • Lipid Bilayers
  • Phosphatidylcholines
  • Protein Aggregates
  • alpha-Synuclein
  • L-Lactate Dehydrogenase
  • 1,2-oleoylphosphatidylcholine