Association of Rituximab Use With Adverse Events in Children, Adolescents, and Young Adults

JAMA Netw Open. 2021 Feb 1;4(2):e2036321. doi: 10.1001/jamanetworkopen.2020.36321.

Abstract

Importance: Rituximab is among the most frequently used immunotherapies in pediatrics. Few studies have reported long-term adverse events associated with its use for children.

Objective: To describe the use of rituximab and to assess whether its use is associated with short- or long-term adverse events, infections, or time to immune reconstitution in a diverse group of young people.

Design, setting, and participants: This retrospective cohort study included 468 patients aged younger than 21 years who received rituximab for diverse indications between October 1, 2010, and December 31, 2017, at Texas Children's Hospital, a large pediatric referral hospital. Patterns of adverse events, infections, and immune recovery are described. Data analyses were conducted from December 2019 to June 2020.

Exposure: One or more doses of rituximab.

Main outcomes and measures: Adverse drug events (eg, anaphylaxis), incidence of mild and severe infections, and time to recovery of B lymphocyte subset counts and immunoglobulin levels. Survival models and logistic regression analyses and were used to identify associated risk factors of infectious and noninfectious adverse drug events.

Results: We identified 468 patients receiving at least 1 dose of rituximab. The total follow-up time was 11 713 person-months. Of the 468 patients, 293 (62.6%) were female, the median (interquartile range) age at receipt of dose was 14.3 (9.9-16.8) years, and 209 (44.7%) were self-reported White Hispanic. Adverse events associated with rituximab infusion occurred in 72 patients (15.4%), and anaphylaxis occurred in 17 patients (3.6%). Long-term adverse events, such as prolonged neutropenia and leukoencephalopathy, were absent. Infections occurred in 224 patients (47.9%); 84 patients (17.9%) had severe infections, and 3 patients (0.6%) had lethal infections. Concurrent use of intravenous chemotherapy, treatment of systemic lupus erythematosus, neutropenia, and use of intravenous immunoglobulin were associated with increased risk of infection. Among 135 patients (28.8%) followed up to B cell count recovery, CD19+ or CD20+ cell numbers normalized in a median of 9.0 months (interquartile range, 5.9-14.4 months) following rituximab use; 48 of 95 patients (51%) evaluated beyond a year had low-for-age B cell counts. Recovery of CD27+ memory B cell number occurred in a median of 15.7 months (interquartile range, 6.0-22.7 months). Among patients with normal baseline values, low immunoglobulin G (IgG) levels developed in 67 of 289 patients (23.2%) and low IgM levels in 118 of 255 patients (40.8%); of these patients evaluated beyond 12 months from rituximab, 16 of 117 (13.7%) had persistently low IgG and 37 (33.9%) of 109 had persistently low IgM.

Conclusions and relevance: Rituximab is well tolerated among young people and is associated with few serious adverse events, but infections are common, corresponding to a prolonged period of B cell count recovery often lasting for longer than a year. Further examination of strategies to prevent infections following rituximab should be pursued.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adolescent
  • Agammaglobulinemia / chemically induced
  • Agammaglobulinemia / epidemiology
  • Anaphylaxis / chemically induced
  • Anaphylaxis / epidemiology*
  • Autoimmune Diseases of the Nervous System / drug therapy
  • B-Lymphocytes
  • Child
  • Child, Preschool
  • Cohort Studies
  • Encephalitis / drug therapy
  • Female
  • Humans
  • Immunoglobulins, Intravenous / therapeutic use
  • Immunologic Factors / adverse effects*
  • Infant
  • Infections / chemically induced
  • Infections / epidemiology*
  • Injection Site Reaction / epidemiology*
  • Leukoencephalopathy, Progressive Multifocal / epidemiology
  • Long Term Adverse Effects / chemically induced
  • Long Term Adverse Effects / epidemiology
  • Lupus Erythematosus, Systemic / drug therapy
  • Lymphocyte Count
  • Lymphoma / drug therapy
  • Male
  • Multiple Sclerosis / drug therapy
  • Nephrotic Syndrome / drug therapy
  • Neutropenia / chemically induced
  • Neutropenia / epidemiology*
  • Odds Ratio
  • Proportional Hazards Models
  • Purpura, Thrombocytopenic, Idiopathic / drug therapy
  • Rituximab / adverse effects*
  • Severity of Illness Index
  • Time Factors
  • Young Adult

Substances

  • Immunoglobulins, Intravenous
  • Immunologic Factors
  • Rituximab