Platelet-expressed immune checkpoint regulator GITRL in breast cancer

Cancer Immunol Immunother. 2021 Sep;70(9):2483-2496. doi: 10.1007/s00262-021-02866-y. Epub 2021 Feb 4.

Abstract

Owing to their key role in several diseases including cancer, activating and inhibitory immune checkpoint molecules are increasingly exploited as targets for immunotherapy. Recently, we demonstrated that platelets, which largely influence tumor progression and immune evasion, functionally express the ligand of the checkpoint molecule GITR. This immunoreceptor modulates effector functions of T cells and NK cells with its function varying dependent on cellular context and activation state. Here, we provide a comparative analysis of platelet-derived GITRL (pGITRL) in breast cancer patients and healthy volunteers. The levels of pGITRL were found to be higher on platelets derived from cancer patients and appeared to be specifically regulated during tumor progression as exemplified by several clinical parameters including tumor stage/grade, the occurrence of metastases and tumor proliferation (Ki67) index. In addition, we report that pGITRL is upregulated during platelet maturation and particularly induced upon exposure to tumor-derived soluble factors. Our data indicate that platelets modulate the GITR/GITRL immune checkpoint in the context of malignant disease and provide a rationale to further study the GITR/GITRL axis for exploitation for immunotherapeutic intervention in cancer patients.

Keywords: Breast cancer; GITRL; Immune checkpoint; Platelets.

MeSH terms

  • Biomarkers, Tumor
  • Blood Platelets / metabolism*
  • Breast Neoplasms / genetics*
  • Breast Neoplasms / metabolism*
  • Breast Neoplasms / pathology
  • Cell Line, Tumor
  • Female
  • Flow Cytometry
  • Gene Expression Regulation, Neoplastic*
  • Glucocorticoid-Induced TNFR-Related Protein / genetics
  • Glucocorticoid-Induced TNFR-Related Protein / metabolism
  • Humans
  • Immune Checkpoint Proteins / genetics*
  • Immune Checkpoint Proteins / metabolism
  • Immunophenotyping
  • Lymphocytes / immunology
  • Lymphocytes / metabolism
  • Odds Ratio
  • Platelet Activation
  • Platelet Aggregation
  • Tumor Necrosis Factors / genetics*
  • Tumor Necrosis Factors / metabolism

Substances

  • Biomarkers, Tumor
  • Glucocorticoid-Induced TNFR-Related Protein
  • Immune Checkpoint Proteins
  • TNFRSF18 protein, human
  • TNFSF18 protein, human
  • Tumor Necrosis Factors