Generally rare but occasionally severe weight gain after switching to an integrase inhibitor in virally suppressed AGEhIV cohort participants

PLoS One. 2021 May 5;16(5):e0251205. doi: 10.1371/journal.pone.0251205. eCollection 2021.

Abstract

Objectives: Recent studies have reported disproportionate weight gain associated with integrase strand transfer inhibitor (INSTI) initiation in antiretroviral therapy(ART)-naive people with HIV (PWH), particularly among black women. We investigated if HIV-positive AGEhIV participants with suppressed viremia switching to INSTI-containing ART experienced more weight gain compared to HIV-positive virally-suppressed non-switching and HIV-negative controls.

Methods: In the AGEhIV cohort, standardized weight measurements were performed biennially. Participants switching to INSTI-containing ART were 1:2:2 propensity score-matched with controls by age, gender, ethnicity and body mass index. Mean weight changes and proportions experiencing >5% or >10% weight gain were compared between study-groups using linear mixed-effects models and logistic regression, respectively.

Results: 121 INSTI-switching participants and 242 participants from each of the control groups were selected. Across groups, median age was 53-55 years, 83-91% were male and 88-93% white. Mean weight change after switch among INSTI-switching participants was +0.14 kg/year (95%CI -0.25, +0.54) and similar among HIV-positive [+0.13 kg/year (95%CI +0.07, +0.33; P = .9)] and HIV-negative [+0.18 kg/year (95%CI 0.00, +0.37; P = .9)] controls. Weight gain >5% occurred in 28 (23.1%) INSTI-switching, 38 HIV-positive (15.7%, P = .085) and 32 HIV-negative controls (13.2%, P = .018). Weight gain >10% was rare.

Conclusions: Switching to INSTI-containing ART in our cohort of predominantly white men on long-term ART was not associated with greater mean weight gain, but >5% weight gain was more common than in controls. These results suggest that not all, but only certain, PWH may be particularly prone to gain a clinically significant amount of weight as a result of switching to INSTI.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Body Mass Index
  • Cohort Studies
  • Female
  • HIV Infections / drug therapy*
  • HIV Infections / physiopathology*
  • HIV Integrase Inhibitors / therapeutic use*
  • Humans
  • Male
  • Middle Aged
  • Weight Gain / drug effects*
  • Weight Gain / physiology*

Substances

  • HIV Integrase Inhibitors

Grants and funding

This work was supported by The Netherlands Organization for Health Research and Development (ZonMW, https://www.zonmw.nl/en/, grant number 300020007) and AIDS Fonds (https://aidsfonds.nl/, grant number 2009063). Additional unrestricted scientific grants were received from Gilead Sciences (https://www.gilead.com/); ViiV Healthcare (https://viivhealthcare.com/en-us/); Janssen Pharmaceuticals N.V. (https://www.janssen.com/); and Merck&Co (https://www.merck.com/). The funders had no role in study design, data collection and analysis, decision to publish, or preparation of the manuscript. All grands were received by PR.