miR-424/503 modulates Wnt/β-catenin signaling in the mammary epithelium by targeting LRP6

EMBO Rep. 2021 Dec 6;22(12):e53201. doi: 10.15252/embr.202153201. Epub 2021 Oct 11.

Abstract

During the female lifetime, the expansion of the epithelium dictated by the ovarian cycles is supported by a transient increase in the mammary epithelial stem cell population (MaSCs). Notably, activation of Wnt/β-catenin signaling is an important trigger for MaSC expansion. Here, we report that the miR-424/503 cluster is a modulator of canonical Wnt signaling in the mammary epithelium. We show that mammary tumors of miR-424(322)/503-depleted mice exhibit activated Wnt/β-catenin signaling. Importantly, we show a strong association between miR-424/503 deletion and breast cancers with high levels of Wnt/β-catenin signaling. Moreover, miR-424/503 cluster is required for Wnt-mediated MaSC expansion induced by the ovarian cycles. Lastly, we show that miR-424/503 exerts its function by targeting two binding sites at the 3'UTR of the LRP6 co-receptor and reducing its expression. These results unveil an unknown link between the miR-424/503, regulation of Wnt signaling, MaSC fate, and tumorigenesis.

Keywords: LRP6; Wnt/β-catenin; breast cancer; miR-424/503.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, Non-P.H.S.

MeSH terms

  • Animals
  • Breast Neoplasms
  • Carcinogenesis
  • Cell Line, Tumor
  • Epithelial Cells / cytology
  • Epithelium* / metabolism
  • Female
  • Low Density Lipoprotein Receptor-Related Protein-6* / genetics
  • Low Density Lipoprotein Receptor-Related Protein-6* / metabolism
  • Mammary Glands, Animal / cytology*
  • Menstrual Cycle
  • Mice
  • MicroRNAs* / genetics
  • Stem Cells / cytology
  • Wnt Signaling Pathway*

Substances

  • Low Density Lipoprotein Receptor-Related Protein-6
  • Lrp6 protein, mouse
  • MIRN424 microRNA, mouse
  • MicroRNAs
  • Mirn503 microRNA, mouse