Effect of ibrutinib with R-CHOP chemotherapy in genetic subtypes of DLBCL

Cancer Cell. 2021 Dec 13;39(12):1643-1653.e3. doi: 10.1016/j.ccell.2021.10.006. Epub 2021 Nov 4.

Abstract

In diffuse large B cell lymphoma (DLBCL), tumors belonging to the ABC but not GCB gene expression subgroup rely upon chronic active B cell receptor signaling for viability, a dependency that is targetable by ibrutinib. A phase III trial ("Phoenix;" ClinicalTrials.gov: NCT01855750) showed a survival benefit of ibrutinib addition to R-CHOP chemotherapy in younger patients with non-GCB DLBCL, but the molecular basis for this benefit was unclear. Analysis of biopsies from Phoenix trial patients revealed three previously characterized genetic subtypes of DLBCL: MCD, BN2, and N1. The 3-year event-free survival of younger patients (age ≤60 years) treated with ibrutinib plus R-CHOP was 100% in the MCD and N1 subtypes while the survival of patients with these subtypes treated with R-CHOP alone was significantly inferior (42.9% and 50%, respectively). This work provides a mechanistic understanding of the benefit of ibrutinib addition to chemotherapy, supporting its use in younger patients with non-GCB DLBCL.

Keywords: ABC DLBCL; BTK inhibitor; CD79B; MYD88; NOTCH1; cancer genomics; memory B cell; precision medicine.

Publication types

  • Research Support, N.I.H., Intramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adenine / analogs & derivatives*
  • Adenine / pharmacology
  • Adenine / therapeutic use
  • Aged
  • Antineoplastic Combined Chemotherapy Protocols / pharmacology
  • Antineoplastic Combined Chemotherapy Protocols / therapeutic use*
  • Cyclophosphamide / pharmacology
  • Cyclophosphamide / therapeutic use
  • Doxorubicin / pharmacology
  • Doxorubicin / therapeutic use
  • Female
  • Humans
  • Lymphoma, Large B-Cell, Diffuse / drug therapy*
  • Male
  • Middle Aged
  • Piperidines / pharmacology
  • Piperidines / therapeutic use*
  • Prednisone / pharmacology
  • Prednisone / therapeutic use
  • Rituximab / pharmacology
  • Rituximab / therapeutic use
  • Vincristine / pharmacology
  • Vincristine / therapeutic use

Substances

  • Piperidines
  • R-CHOP protocol
  • ibrutinib
  • Rituximab
  • Vincristine
  • Doxorubicin
  • Cyclophosphamide
  • Adenine
  • Prednisone

Associated data

  • ClinicalTrials.gov/NCT01855750