Single-Particle Resolution of Copper-Associated Annular α-Synuclein Oligomers Reveals Potential Therapeutic Targets of Neurodegeneration

ACS Chem Neurosci. 2022 May 4;13(9):1410-1421. doi: 10.1021/acschemneuro.2c00021. Epub 2022 Apr 12.

Abstract

Metal ions stabilize protein-protein interactions and can modulate protein aggregation. Here, using liquid-based atomic force microscopy and molecular dynamics simulations, we study the concentration-dependent effect of Cu2+ ions on the aggregation pathway of α-synuclein (α-Syn) proteins, which play a key role in the pathology of Parkinson's disease. The full spectrum of α-Syn aggregates in the presence and absence of Cu2+ ions from monomers to mature fibrils was resolved and quantified at the gold-water interface. Raman spectroscopy confirmed the atomic force microscopy (AFM) findings on the heterogeneity in aggregated states of α-Syn. The formation of annular oligomers was exclusively detected upon incubating α-Syn with Cu2+ ions. Our findings emphasize the importance of targeting annular α-Syn protein oligomers for therapeutic intervention and their potential role as biomarkers for early detection and monitoring progression of neurodegeneration.

Keywords: Raman spectroscopy; atomic force microscopy; metal−protein interactions; molecular dynamics simulations; neurodegeneration; peptide self-assembly.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Copper
  • Humans
  • Microscopy, Atomic Force
  • Parkinson Disease* / metabolism
  • Protein Aggregates
  • alpha-Synuclein* / metabolism

Substances

  • Protein Aggregates
  • alpha-Synuclein
  • Copper