Ornithine Aspartate and Vitamin-E Combination Has Beneficial Effects on Cardiovascular Risk Factors in an Animal Model of Nonalcoholic Fatty Liver Disease in Rats

Biomolecules. 2022 Nov 28;12(12):1773. doi: 10.3390/biom12121773.

Abstract

Cardiovascular (CV) disease is the main cause of death in nonalcoholic fatty liver disease (NAFLD), a clinical condition without any approved pharmacological therapy. Thus, we investigated the effects of ornithine aspartate (LOLA) and/or Vitamin E (VitE) on CV parameters in a steatohepatitis experimental model. Adult Sprague Dawley rats were randomly assigned (10 animals each) and treated from 16 to 28 weeks with gavage as follows: controls (standard diet plus distilled water (DW)), NAFLD (high-fat choline-deficient diet (HFCD) plus DW), NAFLD+LOLA (HFCD plus LOLA (200 mg/kg/day)), NAFLD+VitE (HFCD plus VitE (150 mg twice a week)) or NAFLD+LOLA+VitE in the same doses. Atherogenic ratios were higher in NAFLD when compared with NAFLD+LOLA+VitE and controls (p < 0.05). Serum concentration of IL-1β, IL-6, TNF-α, MCP-1, e-selectin, ICAM-1, and PAI-1 were not different in intervention groups and controls (p > 0.05). NAFLD+LOLA decreased miR-122, miR-33a, and miR-186 (p < 0.05, for all) in relation to NAFLD. NAFLD+LOLA+VitE decreased miR-122, miR-33a and miR-186, and increased miR-126 (p < 0.05, for all) in comparison to NAFLD and NAFLD+VitE. NAFLD+LOLA and NAFLD+LOLA+VitE prevented liver collagen deposition (p = 0.006) in comparison to NAFLD. Normal cardiac fibers (size and shape) were lower in NAFLD in relation to the others; and the inverse was reported for the percentage of regular hypertrophic cardiomyocytes. NAFLD+LOLA+VitE promoted a significant improvement in atherogenic dyslipidemia, liver fibrosis, and paracrine signaling of lipid metabolism and endothelial dysfunction. This association should be further explored in the treatment of NAFLD-associated CV risk factors.

Keywords: animal model; cardiovascular risk; nonalcoholic fatty liver disease; ornithine aspartate; steatohepatitis; vitamin E.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Cardiovascular Diseases* / drug therapy
  • Cardiovascular Diseases* / metabolism
  • Dipeptides* / therapeutic use
  • Disease Models, Animal
  • Drug Therapy, Combination
  • Liver / metabolism
  • MicroRNAs / metabolism
  • Non-alcoholic Fatty Liver Disease* / complications
  • Rats
  • Rats, Sprague-Dawley
  • Risk Factors
  • Vitamin E* / therapeutic use

Substances

  • MicroRNAs
  • ornithylaspartate
  • Vitamin E
  • Dipeptides

Grants and funding

This study was supported by the following Brazilian funding agencies: Biolab Sanus Farmacêutica; National Council for Scientific and Technological Development, CNPq; Coordination for the Improvement of Higher Education Personnel, CAPES/PNPD and Research Incentive Fund from Hospital de Clínicas de Porto Alegre, FIPE-HCPA.