Pharmacokinetics of ciprofloxacin in the elderly

Respiration. 1987;51(4):292-5. doi: 10.1159/000195216.

Abstract

The pharmacokinetics of ciprofloxacin, administered orally as a 250-mg tablet were compared in 10 young (age 20-30 years) and 10 elderly (age 60-73 years) healthy volunteers. The time to peak serum concentrations was about 80 min in both age groups, although the maximum concentration attained was significantly greater in the old (1.7 mg/l) than the young (1.2 mg/l). Area under the plasma concentration-time curve, corrected for body weight, was on average 48% greater in the elderly, but the mean terminal elimination half-life was not significantly different, averaging 4.3 h in the old and 3.7 h in the young. Overall 24-hour urinary recovery in both age groups was comparable. The differences may be explained by a reduced volume of distribution of ciprofloxacin in old age and do not suggest a general need for significant dose alteration in the elderly.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Administration, Oral
  • Adult
  • Aged
  • Aging / metabolism*
  • Biological Availability
  • Ciprofloxacin / blood
  • Ciprofloxacin / pharmacokinetics*
  • Ciprofloxacin / urine
  • Female
  • Half-Life
  • Humans
  • Male
  • Middle Aged

Substances

  • Ciprofloxacin