Cyanotoxin exposure and hepatocellular carcinoma

Toxicology. 2023 Mar 15:487:153470. doi: 10.1016/j.tox.2023.153470. Epub 2023 Feb 28.

Abstract

Cyanobacteria are ubiquitous in aquatic and terrestrial environments worldwide and include a number of species producing tumor-promoting hepatotoxins. Human exposure to cyanobacteria and cyanotoxins primarily occurs though ingestion of contaminated drinking water and food sources. In a Northeast U.S. population, we recently reported an independent association of oral cyanobacteria with risk of hepatocellular carcinoma (HCC). In a cross-sectional study of 55 HCC patients in Hawaii, U.S.A., serum microcystin/nodularin (MC/NOD), cylindrospermopsin (CYN), and anabaenopeptin (AB) were measured by ELISA. In a subset of 16 patients, cyanotoxin levels were compared by tumor expression of over 700 genes analyzed via the Nanostring nCounter Fibrosis panel. MC/NOD, CYN, and AB were detected in all HCC patients. MC/NOD and CYN levels significantly varied by etiology with the highest levels in cases attributed to metabolic risk factors, specifically, hyperlipidemia, type 2 diabetes, and non-alcoholic fatty liver disease/non-alcoholic steatohepatitis. Cyanotoxin levels were significantly positively correlated with tumor expression of genes functioning in PPAR signaling and lipid metabolism. Our study provides novel albeit limited evidence that cyanotoxins may a role in the pathogenesis of HCC through the dysregulation of lipid metabolism and progression of hepatic steatosis.

Keywords: Cancer; Cyanotoxins; Cylindrospermopsin; Liver; Microcystin; Nodularin.

Publication types

  • Research Support, N.I.H., Extramural

MeSH terms

  • Bacterial Toxins* / toxicity
  • Carcinoma, Hepatocellular* / chemically induced
  • Cross-Sectional Studies
  • Cyanobacteria Toxins
  • Cyanobacteria* / metabolism
  • Diabetes Mellitus, Type 2*
  • Humans
  • Liver Neoplasms* / chemically induced
  • Marine Toxins
  • Microcystins / toxicity

Substances

  • Bacterial Toxins
  • Marine Toxins
  • Cyanobacteria Toxins
  • Microcystins