IL16 and factor V gene variations are associated with asparaginase-related thrombosis in childhood acute lymphoblastic leukemia patients

Pharmacogenomics. 2023 Mar;24(4):199-206. doi: 10.2217/pgs-2022-0164. Epub 2023 Mar 22.

Abstract

Aim: We previously conducted exome-wide association study in acute lymphoblastic leukemia patients and identified association of five SNPs with asparaginase-related thrombosis. Here we aimed to replicate these findings in an independent patient cohort and through analyses in vitro. Patients & methods: SNPs located in IL16, MYBBP1A, PKD2L1, RIN3 and MPEG1 genes were analyzed in patients receiving Dana-Farber Cancer Institute acute lymphoblastic leukemia treatment protocols 05-001 and 11-001. Thrombophilia-related variations were also analysed. Results: IL16 rs11556218 conferred higher risk of thrombosis and higher in vitro sensitivity to asparaginase. The association was modulated by the treatment protocol, risk group and immunophenotype. A crosstalk between factor V Leiden, non-O blood groups and higher risk of thrombosis was also seen. Conclusion: IL16 and factor V Leiden variations are implicated in asparaginase-related thrombosis.

Keywords: FVL; IL16; acute lymphoblastic leukemia; asparaginase; lymphoblastoid cell lines; pharmacogenetics; single nucleotide polymorphism; thrombosis.

Plain language summary

This study looked at how certain genetic variations are related to a higher risk of blood clots in children with a type of cancer called acute lymphoblastic leukemia who are receiving a certain treatment (asparaginase). The study found that one specific genetic variation (IL16 rs11556218) was linked to a higher risk of blood clots (thrombosis), and that this risk was influenced by disease and treatment features. The study also found that a certain genetic variation (factor V Leiden), which makes blood more likely to clot, and blood type (non-O) were linked to a higher risk of thrombosis. The conclusion of this study is that genetic variations may play a role in blood clots in children with acute lymphoblastic leukemia receiving asparaginase, and if further confirmed, these variations can serve to advance personalized treatment strategies.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Antineoplastic Agents* / therapeutic use
  • Asparaginase / adverse effects
  • Calcium Channels
  • DNA-Binding Proteins
  • Factor V / genetics
  • Factor V / therapeutic use
  • Humans
  • Interleukin-16 / therapeutic use
  • Precursor Cell Lymphoblastic Leukemia-Lymphoma* / complications
  • Precursor Cell Lymphoblastic Leukemia-Lymphoma* / drug therapy
  • Precursor Cell Lymphoblastic Leukemia-Lymphoma* / genetics
  • RNA-Binding Proteins
  • Receptors, Cell Surface
  • Thrombosis* / chemically induced
  • Thrombosis* / genetics
  • Transcription Factors

Substances

  • Asparaginase
  • Interleukin-16
  • Antineoplastic Agents
  • Factor V
  • MYBBP1A protein, human
  • DNA-Binding Proteins
  • Transcription Factors
  • RNA-Binding Proteins
  • PKD2L1 protein, human
  • Receptors, Cell Surface
  • Calcium Channels