Engineering a potent boron-10-enriched polymeric nanoparticle for boron neutron capture therapy

Nanomedicine (Lond). 2023 Apr;18(9):743-754. doi: 10.2217/nnm-2022-0330. Epub 2023 Jun 12.

Abstract

Background: Boron neutron capture therapy (BNCT) is a promising cancer treatment that eliminates tumor cells by triggering high-energy radiation within cancer cells. Aim: In vivo evaluation of poly(vinyl alcohol)/boric acid crosslinked nanoparticles (PVA/BA NPs) for BNCT. Materials & methods: PVA/BA NPs were synthesized and intravenously injected into tumor-bearing mice for BNCT. Results: The in vitro boron uptake of PVA/BA NPs in tumor cells was 70-fold higher than the required boron uptake for successful BNCT. In an in vivo study, PVA/BA NPs showed a 44.29% reduction in tumor size compared with clinically used boronophenylalanine for oral cancer in a murine model. Conclusion: PVA/BA NPs exhibited effective therapeutic results for oral cancer treatments in BNCT.

Keywords: BNCT; boric acid; head and neck cancer; poly(vinyl alcohol); polymeric nanoparticles.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Boron Neutron Capture Therapy* / methods
  • Chemical Engineering
  • Disease Models, Animal
  • Male
  • Mice
  • Mouth Neoplasms* / radiotherapy
  • Nanoparticles*

Substances

  • Boron-10