Effects of storage up to 1 year on the in vitro antimicrobial activity of preformulated antibiotic-impregnated calcium sulfate beads

Vet Surg. 2024 Jul;53(5):918-925. doi: 10.1111/vsu.14014. Epub 2023 Aug 13.

Abstract

Objective: To compare antimicrobial activity as demonstrated by the zone of inhibition (ZOI) produced by antibiotic-impregnated calcium sulfate (CaSO4) beads after storage for 0, 3, 6, 9, and 12 months.

Study design: Controlled laboratory study.

Sample population: Three-millimeter diameter CaSO4 beads impregnated with vancomycin (125 mg/mL), or amikacin (250 mg/mL), or without antibiotic (control).

Methods: Calcium sulfate beads were created at the onset of the study. Individual beads were separated in sterile containers and stored in a closed cabinet at room temperature and humidity for 0, 3, 6, 9, or 12 months until testing. The ZOI against methicillin-resistant Staphylococcus pseudintermedius, methicillin-resistant Staphylococcus aureus, and Pseudomonas aeruginosa was recorded with serial replating on a fresh lawn of bacteria every 24 h until beads failed to produce a ZOI. The ZOIs and their changes were compared with mixed-effects linear models. Eluted concentrations of vancomycin measured with high-performance liquid chromatography were reported.

Results: At 24 h, ZOIs were comparable regardless of time since formulation, except vancomycin against P. aeruginosa, which failed to generate a ZOI. The daily changes of ZOI and duration of activity of antibiotics did not vary between storage length (p > .05). There was no consistent change in eluted drug concentration between storage length of beads.

Conclusion: Light protected storage at room temperature for up to 12 months did not impair the in vitro activity of antibiotic-impregnated CaSO4 beads, as demonstrated through ZOIs.

Clinical significance: When stored correctly, antibiotic-impregnated CaSO4 beads can be used at least up to 12 months after formulation.

MeSH terms

  • Amikacin / administration & dosage
  • Amikacin / pharmacology
  • Anti-Bacterial Agents* / administration & dosage
  • Anti-Bacterial Agents* / chemistry
  • Anti-Bacterial Agents* / pharmacology
  • Calcium Sulfate* / chemistry
  • Calcium Sulfate* / pharmacology
  • Drug Stability
  • Drug Storage*
  • Methicillin-Resistant Staphylococcus aureus / drug effects
  • Microbial Sensitivity Tests
  • Pseudomonas aeruginosa* / drug effects
  • Time Factors
  • Vancomycin* / chemistry
  • Vancomycin* / pharmacology

Substances

  • Calcium Sulfate
  • Anti-Bacterial Agents
  • Vancomycin
  • Amikacin