Real-World Patient Experience of Pexidartinib for Tenosynovial Giant-Cell Tumor

Oncologist. 2024 Apr 4;29(4):e535-e543. doi: 10.1093/oncolo/oyad282.

Abstract

Background: Pexidartinib (Turalio) is the only systemic therapy approved by the FDA for the treatment of adult patients with symptomatic tenosynovial giant-cell tumor (TGCT) associated with severe morbidity or functional limitations, and not amenable to improvement with surgery. This study assessed patient-reported treatment experiences and symptom improvement among patients receiving pexidartinib.

Methods: A cross-sectional, web-based survey collected data on demographics, disease history, pexidartinib dosing, and symptoms before and after pexidartinib use.

Results: Of 288 patients enrolled in the Turalio REMS program in May 2021, 83 completed the survey: mean age was 44.2 years, 62.7% were female, and most common tumor sites were in knee (61%) and ankle (12%). Mean initial dose was 622 mg/day: 29 patients reported reduction from initial dose and 8 had dose reduction after titrating up to a higher dose. At the time of survey completion, median time on pexidartinib was 6.0 months; 22 (26.5%) patients discontinued pexidartinib due to physician suggestion, abnormal laboratory results, side effect, or symptom improvement. Compared with before pexidartinib initiation, most patients reported improvement in overall TGCT symptom (78.3%) and physical function (77.2%) during pexidartinib treatment. Significant improvement was reported during pexidartinib treatment in worst stiffness numeric rating scale (NRS) (3.0 vs. 6.2, P < .05) and worst pain NRS (2.7 vs. 5.7, P < .05).

Conclusion: Findings from this cross-sectional survey confirmed the benefit of pexidartinib in improving symptoms and functional outcomes among patients with symptomatic TGCTs from the patients' perspective. Future research is warranted to examine the long-term benefit and risk of pexidartinib.

Keywords: patient-reported outcome; pexidartinib; symptom change; tenosynovial giant-cell tumor.

MeSH terms

  • Adult
  • Aminopyridines / therapeutic use
  • Cross-Sectional Studies
  • Female
  • Giant Cell Tumor of Tendon Sheath* / drug therapy
  • Giant Cell Tumor of Tendon Sheath* / pathology
  • Giant Cell Tumor of Tendon Sheath* / surgery
  • Humans
  • Male
  • Patient Outcome Assessment
  • Pyrroles*

Substances

  • pexidartinib
  • Aminopyridines
  • Pyrroles