KIO3-catalyzed selective oxidation of thiols to disulfides in water under ambient conditions

Org Biomol Chem. 2024 Mar 13;22(11):2175-2181. doi: 10.1039/d3ob01913f.

Abstract

Herein, we report a KIO3-catalyzed oxidative coupling of thiols to their corresponding disulfides in water, in a short time and at ambient temperature. The reaction has a broad scope and exhibits good functional group tolerance, resulting in the desired products in excellent yields. This approach allows the reuse of the reaction system in multiple cycles and scale-up. Furthermore, the current protocol demonstrates compatibility for in situ generation of disulfides and post application in C(sp2)-H bond sulfenylation.