CYP7B1-mediated 25-hydroxycholesterol degradation maintains quiescence-activation balance and improves therapeutic potential of mesenchymal stem cells

Cell Chem Biol. 2024 Jul 18;31(7):1277-1289.e7. doi: 10.1016/j.chembiol.2024.01.009. Epub 2024 Feb 20.

Abstract

Stem cells remain quiescent in vivo and become activated in response to external stimuli. However, the mechanism regulating the quiescence-activation balance of bone-marrow-derived mesenchymal stem cells (BM-MSCs) is still unclear. Herein, we demonstrated that CYP7B1 was the common critical molecule that promoted activation and impeded quiescence of BM-MSCs under inflammatory stimulation. Mechanistically, CYP7B1 degrades 25-hydroxycholesterol (25-HC) into 7α,25-dihydroxycholesterol (7α,25-OHC), which alleviates the quiescence maintenance effect of 25-HC through Notch3 signaling pathway activation. CYP7B1 expression in BM-MSCs was regulated by NF-κB p65 under inflammatory conditions. BM-MSCs from CYP7B1 conditional knockout (CKO) mice had impaired activation abilities, relating to the delayed healing of bone defects. Intravenous infusion of BM-MSCs overexpressing CYP7B1 could improve the pathological scores of mice with collagen-induced arthritis. These results clarified the quiescence-activation regulatory mechanism of BM-MSCs through the NF-κB p65-CYP7B1-Notch3 axis and provided insight into enhancing BM-MSCs biological function as well as the subsequent therapeutic effect.

Keywords: 25-hydroxycholesterol; CYP7B1; Notch3; mesenchymal stem cells; quiescence.

MeSH terms

  • Animals
  • Arthritis, Experimental / metabolism
  • Arthritis, Experimental / pathology
  • Cells, Cultured
  • Cytochrome P450 Family 7* / metabolism
  • Humans
  • Hydroxycholesterols* / metabolism
  • Hydroxycholesterols* / pharmacology
  • Male
  • Mesenchymal Stem Cell Transplantation
  • Mesenchymal Stem Cells* / cytology
  • Mesenchymal Stem Cells* / metabolism
  • Mice
  • Mice, Inbred C57BL*
  • Mice, Knockout*
  • Receptor, Notch3 / genetics
  • Receptor, Notch3 / metabolism
  • Signal Transduction / drug effects
  • Steroid Hydroxylases
  • Transcription Factor RelA / metabolism

Substances

  • 25-hydroxycholesterol
  • Cyp7b1 protein, mouse
  • Cytochrome P450 Family 7
  • Hydroxycholesterols
  • Receptor, Notch3
  • Steroid Hydroxylases
  • Transcription Factor RelA
  • CYP7B1 protein, human