Recent Advances in Metal-Catalyzed Approaches for the Synthesis of Quinazoline Derivatives

Molecules. 2024 May 16;29(10):2353. doi: 10.3390/molecules29102353.

Abstract

Quinazolines are an important class of heterocyclic compounds that have proven their significance, especially in the field of organic synthesis and medicinal chemistry because of their wide range of biological and pharmacological properties. Thus, numerous synthetic methods have been developed for the synthesis of quinazolines and their derivatives. This review article briefly outlines the new synthetic methods for compounds containing the quinazoline scaffold employing transition metal-catalyzed reactions.

Keywords: C-H activation; cascade reactions; intramolecular dehydrative/dehydrogenative cyclizations; quinazoline heterocycles; transition metal-catalyzed synthesis.

Publication types

  • Review

Grants and funding

J.M.S. acknowledges different grant for support P30 CA010815, S10 OD030245, P01 CA114046, P01 CA269043, R01 CA272645.