STAT3 Regulates the Redox Profile in MDA-MB-231 Breast Cancer Cells

Cell Biochem Biophys. 2024 Dec;82(4):3507-3516. doi: 10.1007/s12013-024-01439-x. Epub 2024 Jul 20.

Abstract

Unbalanced redox status and constitutive STAT3 activation are related to several aspects of tumor biology and poor prognosis, including metastasis and drug resistance. The triple-negative breast cancer (TNBC) is listed as the most aggressive and exhibits the worst prognosis among the breast cancer subtypes. Although the mechanism of reactive oxygen species (ROS) generation led to STAT3 activation is described, there is no data concerning the STAT3 influence on redox homeostasis in TNBC. To address the role of STAT3 signaling in redox balance, we inhibited STAT3 in TNBC cells and investigated its impact on total ROS levels, contents of hydroperoxides, nitric oxide (NO), and total glutathione (GSH), as well as the expression levels of 3-nitrotyrosine (3NT), nuclear factor (erythroid-derived 2)-like 2 (Nrf2), and nuclear factor kappa B (NF-κB)/p65. Our results indicate that ROS levels depend on the STAT3 activation, while the hydroperoxide level remained unchanged, and NO and 3NT expression increased. Furthermore, GSH levels, Nrf2, and NF-κB/p65 protein levels are decreased in the STAT3-inhibited cells. Accordingly, TNBC patients' data from TCGA demonstrated that both STAT3 mRNA levels and STAT3 signature are correlated to NF-κB/p65 and Nrf2 signatures. Our findings implicate STAT3 in controlling redox balance and regulating redox-related genes' expression in triple-negative breast cancer.

Keywords: Breastcancer; Redox; STAT3; TNBC.

MeSH terms

  • Cell Line, Tumor
  • Female
  • Glutathione* / metabolism
  • Humans
  • NF-E2-Related Factor 2* / genetics
  • NF-E2-Related Factor 2* / metabolism
  • Nitric Oxide / metabolism
  • Oxidation-Reduction*
  • Reactive Oxygen Species* / metabolism
  • STAT3 Transcription Factor* / metabolism
  • Signal Transduction
  • Transcription Factor RelA / metabolism
  • Triple Negative Breast Neoplasms* / metabolism
  • Triple Negative Breast Neoplasms* / pathology
  • Tyrosine / analogs & derivatives
  • Tyrosine / metabolism

Substances

  • STAT3 Transcription Factor
  • Glutathione
  • Reactive Oxygen Species
  • NF-E2-Related Factor 2
  • Nitric Oxide
  • NFE2L2 protein, human
  • Tyrosine
  • 3-nitrotyrosine
  • Transcription Factor RelA
  • STAT3 protein, human