The Potential of Metabolomics to Find Proper Biomarkers for Addressing the Neuroprotective Efficacy of Drugs Aimed at Delaying Parkinson's and Alzheimer's Disease Progression

Cells. 2024 Jul 31;13(15):1288. doi: 10.3390/cells13151288.

Abstract

The first objective is to highlight the lack of tools to measure whether a given intervention affords neuroprotection in patients with Alzheimer's or Parkinson's diseases. A second aim is to present the primary outcome measures used in clinical trials in cohorts of patients with neurodegenerative diseases. The final aim is to discuss whether metabolomics using body fluids may lead to the discovery of biomarkers of neuroprotection. Information on the primary outcome measures in clinical trials related to Alzheimer's and Parkinson's disease registered since 2018 was collected. We analysed the type of measures selected to assess efficacy, not in terms of neuroprotection since, as stated in the aims, there is not yet any marker of neuroprotection. Proteomic approaches using plasma or CSF have been proposed. PET could estimate the extent of lesions, but disease progression does not necessarily correlate with a change in tracer uptake. We propose some alternatives based on considering the metabolome. A new opportunity opens with metabolomics because there have been impressive technological advances that allow the detection, among others, of metabolites related to mitochondrial function and mitochondrial structure in serum and/or cerebrospinal fluid; some of the differentially concentrated metabolites can become reliable biomarkers of neuroprotection.

Keywords: biomarkers; cognition test; neurodegenerative diseases; neuroprotection; primary outcome measure; protein aggregation.

Publication types

  • Review

MeSH terms

  • Alzheimer Disease* / blood
  • Alzheimer Disease* / drug therapy
  • Alzheimer Disease* / physiopathology
  • Animals
  • Biomarkers* / blood
  • Clinical Trials as Topic
  • Disease Progression
  • Metabolomics*
  • Neuroprotection
  • Parkinson Disease* / blood
  • Parkinson Disease* / drug therapy
  • Parkinson Disease* / physiopathology
  • Proteomics

Substances

  • Biomarkers

Grants and funding

C.G. received from the Ministry of Science and Innovation (MCIN) of Spain an FPI (“Formación de Personal Investigador”) predoctoral contract associated with the PID2021-126600OB-I00 grant (funded by Spanish MCIN/AEI/10.13039/501100011033 and, as appropriate, by “ERDF A way of making Europe”, by the “European Union” or by the “European Union Next Generation EU/PRTR”).