Topology-selective photo-crosslinking of G-quadruplexes via dual G-quartet and groove recognition

Chem Commun (Camb). 2024 Nov 14;60(92):13550-13553. doi: 10.1039/d4cc04804k.

Abstract

The novel photo-crosslinking ligand 6OTD-Bp, bearing an alkylamine benzophenone (Bp) with macrocyclic hexaoxazole (6OTD), was shown to preferentially ligate with hybrid G4s through recognizing both G-quartets and their characteristic wide groove. Higher crosslinking yield was observed for hybrid G4 with wider grooves.

MeSH terms

  • Benzophenones* / chemistry
  • Cross-Linking Reagents / chemistry
  • G-Quadruplexes*
  • Ligands
  • Molecular Structure
  • Oxazoles / chemistry
  • Photochemical Processes

Substances

  • Benzophenones
  • benzophenone
  • Ligands
  • Cross-Linking Reagents
  • Oxazoles