Delineation of fucosyltransferase activities with thiol reagents

Biochem J. 1979 Sep 1;181(3):767-9. doi: 10.1042/bj1810767.

Abstract

The thiol reagent dithiothreitol inhibits the activity of a core GDP-fucose-N-acetylglucosaminide alpha-6-fucosyltransferase in plasma and blood-cell homogenates, while promoting the activity of alpha-2- and alpha-3-fucosyltransferases. The latter enzymes catalyse transfer of fucose on to terminal galactose and subterminal N-acetylglucosamine residues respectively. A thiol-blocking reagent N-ethylmaleimide does not affect the activity of the alpha-6-fucosyltransferase, but inhibits the other two enzymes. These results indicate the presence of a critical disulphide linkage in the alpha-6-fucosyltransferase, and provide a means of delineation of different fucosyltransferases.

MeSH terms

  • Chemical Phenomena
  • Chemistry
  • Dithiothreitol / pharmacology*
  • Ethylmaleimide / pharmacology*
  • Fucosyltransferases / antagonists & inhibitors*
  • Fucosyltransferases / blood
  • Hexosyltransferases / antagonists & inhibitors*
  • Humans
  • Leukemia / enzymology

Substances

  • Fucosyltransferases
  • Hexosyltransferases
  • Ethylmaleimide
  • Dithiothreitol