Lack of effect of ranitidine on warfarin action

Br J Clin Pharmacol. 1981 Dec;12(6):791-4. doi: 10.1111/j.1365-2125.1981.tb01308.x.

Abstract

1 In five volunteers taking daily subtherapeutic doses of warfarin the addition of ranitidine 200 mg twice daily for 14 days did not affect prothrombin time or plasma warfarin concentration. 2 Ranitidine had no effect on the single dose pharmacodynamics and pharmacokinetics of warfarin in the rat. 3 Ranitidine had no effect on pentobarbitone sleeping time in the rat whereas cimetidine significantly prolonged the sleeping time. 4 The interaction between cimetidine and oral anticoagulants is unrelated to histamine H2-receptor antagonism.

MeSH terms

  • Adult
  • Animals
  • Drug Interactions
  • Furans / pharmacology*
  • Half-Life
  • Histamine H2 Antagonists / pharmacology*
  • Humans
  • Kinetics
  • Male
  • Pentobarbital / pharmacology
  • Prothrombin Time
  • Ranitidine
  • Rats
  • Rats, Inbred Strains
  • Sleep / drug effects
  • Time Factors
  • Warfarin / blood
  • Warfarin / pharmacology*

Substances

  • Furans
  • Histamine H2 Antagonists
  • Warfarin
  • Ranitidine
  • Pentobarbital