Origin of malondialdehyde from DNA degraded by Fe(II) x bleomycin

J Biol Chem. 1980 Dec 25;255(24):11832-8.

Abstract

Ferrous bleomycin is known to break DNA efficiently in vitro in the presence of O2, giving rise to ologonucleotides, bases, and compounds resembling malondialdehyde in their chromogenic reaction with 2-thiobarbituric acid. Chromatography of radiolabeled DNA reaction mixtures resolves three kinds of malondialdehyde-like products, related by sequential conversions. The first chromogenic product is linked to DNA, and its formation does not entail the release of a base. It decomposes readily to the second product, a compound containing the base and deoxyribose carons 1'-3'. Hydrolysis of either product yields the third, which is indistinguishable from authentic malondialdehyde. These findings suggest that the oxygen-dependent cleavage of DNA by Fe(II) x bleomycin can begin with the rupture of the deoxyribose 3'-4'-carbon bond. The initiation of these events is concurrent with the initiation of another mode of DNA degradation, involving the release of free base alone, in a yield similar to that of chromogen.

Publication types

  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Bacteriophage lambda
  • Bleomycin*
  • Chemical Phenomena
  • Chemistry
  • DNA, Viral*
  • Drug Stability
  • Iron*
  • Malonates*
  • Malondialdehyde*
  • Oxidation-Reduction
  • Spectrophotometry

Substances

  • DNA, Viral
  • Malonates
  • Bleomycin
  • Malondialdehyde
  • Iron