Effects of dilazep on human platelets and rat vascular tissue: in vitro studies on platelet aggregation, and arachidonic acid oxidation

Pharmacol Res Commun. 1983 Jun;15(6):593-602. doi: 10.1016/s0031-6989(83)80030-7.

Abstract

The "in vitro" effects of Dilazep on platelet aggregation and arachidonic acid oxidation in platelets and vessel wall were studied. Dilazep exerted a clearcut inhibitory effect on platelet aggregation induced by several stimuli. In addition, the compound completely suppressed malondialdehyde production by platelets elicited by collagen and thrombin, in a dose-dependent fashion. The evaluation of Dilazep effects on the in vitro release of prostacyclin-like material by rat aortic tissue did not provide any indication about an interference of the drug on the generation of endogenous antiaggregatory material.

MeSH terms

  • Animals
  • Aorta / metabolism
  • Arachidonic Acid
  • Arachidonic Acids / metabolism*
  • Azepines / pharmacology*
  • Blood Platelets / drug effects*
  • Blood Platelets / metabolism
  • Blood Vessels / drug effects*
  • Blood Vessels / metabolism
  • Dilazep / pharmacology*
  • Epoprostenol / metabolism
  • Humans
  • In Vitro Techniques
  • Male
  • Malondialdehyde / metabolism
  • Oxidation-Reduction
  • Platelet Aggregation / drug effects
  • Rats

Substances

  • Arachidonic Acids
  • Azepines
  • Arachidonic Acid
  • Malondialdehyde
  • Epoprostenol
  • Dilazep