Characterization of a 60-kilodalton substrate of the insulin receptor kinase

J Biol Chem. 1994 Apr 15;269(15):11498-502.

Abstract

A 60-kDa tyrosine-phosphorylated protein has been observed after insulin treatment of cells in immunoprecipitations of the GTPase-activating protein of Ras (called GAP) as well as the phosphatidylinositol 3-kinase. In the present studies, these two 60-kDa proteins have been shown to differ by limited proteolytic digestions as well as by immunoprecipitation with a monoclonal antibody. This monoclonal antibody was also utilized to show that the 60-kDa GAP-associated protein was rapidly phosphorylated in intact cells after insulin stimulation and to associate with GAP only after insulin treatment of the cells. In addition, the 60-kDa protein was found to be phosphorylated in vitro by the insulin receptor. Finally, the 60-kDa protein immunoprecipitated by this antibody was found not to react with a polyclonal antibody directed against a 62-kDa tyrosine-phosphorylated GAP-associated protein previously observed in src-transformed cells. These studies indicate that insulin stimulates the tyrosine phosphorylation of at least two distinct 60-kDa proteins, one that becomes associated with GAP and appears to be a direct substrate of the insulin receptor kinase and another that associates with the phosphatidylinositol 3-kinase.

Publication types

  • Comparative Study
  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Animals
  • Antibodies, Monoclonal
  • CHO Cells
  • Cricetinae
  • Cross Reactions
  • Electrophoresis, Polyacrylamide Gel
  • GTPase-Activating Proteins
  • Humans
  • Insulin / pharmacology
  • Kinetics
  • Molecular Weight
  • Phosphotyrosine
  • Proteins / isolation & purification
  • Proteins / metabolism
  • Receptor, Insulin / isolation & purification
  • Receptor, Insulin / metabolism*
  • Substrate Specificity
  • Transfection
  • Tyrosine / analogs & derivatives*
  • Tyrosine / isolation & purification
  • Tyrosine / metabolism
  • ras GTPase-Activating Proteins

Substances

  • Antibodies, Monoclonal
  • GTPase-Activating Proteins
  • Insulin
  • Proteins
  • ras GTPase-Activating Proteins
  • Phosphotyrosine
  • Tyrosine
  • Receptor, Insulin