Retrobulbar arterial hemodynamic effects of betaxolol and timolol in normal-tension glaucoma

Am J Ophthalmol. 1995 Aug;120(2):168-75. doi: 10.1016/s0002-9394(14)72604-2.

Abstract

Purpose: beta-Adrenergic blocking drugs lower intraocular pressure. The question of whether these drugs also alter, either directly or indirectly, orbital hemodynamics is potentially of great importance for patients with normal-tension glaucoma who may have some degree of reversible vasospasm.

Methods: We compared the effect of selective (betaxolol) and nonselective (timolol) beta-adrenergic blocking drugs on flow velocities (as determined by color Doppler imaging) in orbital vessels in 13 patients with normal-tension glaucoma (mean age, 62 +/- 3 years; mean intraocular pressure, 15 +/- 2 mm Hg). A one-month drug treatment double-masked crossover design, with a three-week washout before each drug, was used.

Results: Neither drug changed peak systolic velocity in any of the four vessels studied (ophthalmic, nasal and temporal posterior ciliary, and central retinal arteries). Additionally, timolol did not alter end-diastolic velocity or resistance index (defined as [peak systolic velocity minus end-diastolic velocity] divided by peak systolic velocity) in any of the vessels measured. In contrast, betaxolol tended to increase end-diastolic velocity and to decrease resistance index: the four-vessel average end-diastolic velocity increased 30% (P = .08), and the four-vessel average resistance index decreased significantly (P = .04). These reductions in resistance index occurred despite that betaxolol, in contrast to timolol, did not significantly decrease intraocular pressure.

Conclusions: These results suggest that, in patients with normal-tension glaucoma, selective beta-adrenergic blockade (betaxolol) may have ocular vasorelaxant effects independent of any influence on intraocular pressure, whereas nonselective blockade (timolol) lowers intraocular pressure without apparently altering orbital hemodynamics.

Publication types

  • Clinical Trial
  • Comparative Study
  • Randomized Controlled Trial
  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Arteries / diagnostic imaging
  • Arteries / drug effects
  • Arteries / physiology
  • Betaxolol / administration & dosage
  • Betaxolol / pharmacology*
  • Blood Flow Velocity
  • Cross-Over Studies
  • Double-Blind Method
  • Female
  • Glaucoma / drug therapy
  • Glaucoma / physiopathology*
  • Hemodynamics / drug effects
  • Hemodynamics / physiology
  • Humans
  • Intraocular Pressure / drug effects
  • Male
  • Middle Aged
  • Ophthalmic Solutions
  • Orbit / blood supply*
  • Orbit / diagnostic imaging
  • Orbit / drug effects
  • Prospective Studies
  • Timolol / administration & dosage
  • Timolol / pharmacology*
  • Ultrasonography, Doppler, Color
  • Vascular Resistance / drug effects

Substances

  • Ophthalmic Solutions
  • Timolol
  • Betaxolol