Influence of K+ channel openers on interferon-gamma dependent immune response in experimental allergic neuritis (EAN)

Autoimmunity. 1994;18(4):233-41. doi: 10.3109/08916939409009524.

Abstract

We examined the influence of the K+ channel opening drugs BRL 38227, pinacidil and diazoxide on cellular immune response and clinical course of experimental allergic neuritis (EAN) actively induced in Lewis rats by bovine peripheral myelin (BPM). T cell functions of EAN lymph node cells were assessed by measurement of proliferation and by counting of interferon-gamma secreting cells (IFN-gamma sc) in response to the specific antigen BPM and the T cell mitogen phytohemagglutinin (PHA). BRL 38227 and diazoxide at concentrations of 10(-5)M-10(-6)M and pinacidil at concentrations of 10(-5)M-10(-7)M enhanced the proliferative response to both BPM and PHA. The number of IFN-gamma sc was suppressed by the K+ channel openers in the same concentration range. There was a tendency of stronger suppression of cultures with high numbers of BPM-reactive IFN-gamma sc than of cultures with low numbers of BPM-reactive IFN-gamma sc. The applied K+ channel openers are primarily acting on ATP-sensitive K+ channels, which have not been found in T cells so far. The drugs may, therefore, exert non-selective effects on conventional voltage- and/or Ca(++)-dependent channels of T cells. A first trial with in vivo administration of 2.5 mg/kg x day of the drugs resulted in more severe neurological deficits in the early phase of EAN with BRL 38227, whereas pinacidil and diazoxide had no significant effects.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Benzopyrans / pharmacology
  • Cromakalim
  • Diazoxide / pharmacology
  • Guanidines / pharmacology
  • Interferon-gamma / metabolism
  • Interferon-gamma / physiology*
  • Ion Channel Gating / drug effects*
  • Lymph Nodes / cytology
  • Lymphocyte Activation / drug effects
  • Neuritis, Autoimmune, Experimental / immunology*
  • Pinacidil
  • Potassium Channels / drug effects*
  • Pyrroles / pharmacology
  • Rats
  • Rats, Inbred Lew

Substances

  • Benzopyrans
  • Guanidines
  • Potassium Channels
  • Pyrroles
  • Cromakalim
  • Pinacidil
  • Interferon-gamma
  • Diazoxide