Functional expression of a rat homologue of the voltage gated either á go-go potassium channel reveals differences in selectivity and activation kinetics between the Drosophila channel and its mammalian counterpart

EMBO J. 1994 Oct 3;13(19):4451-8. doi: 10.1002/j.1460-2075.1994.tb06767.x.

Abstract

We have cloned a mammalian (rat) homologue of Drosophila ether á go-go (eag) cDNA, which encodes a distinct type of voltage activated potassium (K) channel. The derived Drosophila and rat eag polypeptides share > 670 amino acids, with a sequence identity of 61%, exhibiting a high degree of similarity at the N-terminus, the hydrophobic core including the pore forming P region and a potential cyclic nucleotide binding site. Rat eag mRNA is specifically expressed in the central nervous system. In the Xenopus oocyte expression system rat eag mRNA gives rise to voltage activated K channels which have distinct properties in comparison with Drosophila eag channels and other voltage activated K channels. Thus, the rat eag channel further extends the known diversity of K channels. Most notably, the kinetics of rat eag channel activation depend strongly on holding membrane potential. Hyperpolarization slows down the kinetics of activation; conversely depolarization accelerates the kinetics of activation. This novel K channel property may have important implications in neural signal transduction allowing neurons to tune their repolarizing properties in response to membrane hyperpolarization.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Amino Acid Sequence
  • Animals
  • Base Sequence
  • DNA, Complementary
  • Drosophila
  • Drosophila Proteins
  • Ether-A-Go-Go Potassium Channels
  • Ion Channel Gating / physiology
  • Male
  • Molecular Sequence Data
  • Nerve Tissue Proteins / physiology
  • Oocytes / metabolism
  • Polymerase Chain Reaction
  • Potassium Channels / biosynthesis
  • Potassium Channels / chemistry
  • Potassium Channels / physiology*
  • RNA, Messenger / analysis
  • Rats
  • Rats, Sprague-Dawley
  • Recombinant Proteins / biosynthesis
  • Sequence Homology, Amino Acid
  • Species Specificity
  • Xenopus laevis

Substances

  • DNA, Complementary
  • Drosophila Proteins
  • Ether-A-Go-Go Potassium Channels
  • Kcnh1 protein, rat
  • Nerve Tissue Proteins
  • Potassium Channels
  • RNA, Messenger
  • Recombinant Proteins
  • eag protein, Drosophila

Associated data

  • GENBANK/Z34264