Rapid and transient thrombin stimulation of phosphatidylinositol 4,5-bisphosphate synthesis but not of phosphatidylinositol 3,4-bisphosphate independent of phospholipase C activation in platelets

FEBS Lett. 1993 Sep 20;330(3):347-51. doi: 10.1016/0014-5793(93)80902-7.

Abstract

When platelets are stimulated by thrombin they immediately undergo inositol lipid hydrolysis via phospholipase C activation. However, subsequently an increased production of phosphatidylinositol 4,5-bisphosphate is observed. Phospholipases C were inhibited by lowering the cytoplasmic free calcium concentration by preincubation with Quin-2-tetra(acetoxymethyl) ester. Aggregation and secretion were also totally suppressed. Under these conditions we observed an increased labeling of phosphatidylinositol 4,5-bisphosphate, indicating a stimulation of inositol lipid kinases, independent of lipid hydrolysis by phospholipase C. Conversely the production of phosphatidylinositol 3,4-bisphosphate was totally abolished. These results suggest a different regulation of the kinases/phosphatases responsible for the production of phosphatidylinositol 4,5-bisphosphate and phosphatidylinositol 3,4-bisphosphate.

MeSH terms

  • Aminoquinolines / pharmacology
  • Blood Platelets / enzymology*
  • Cells, Cultured
  • Enzyme Activation
  • Humans
  • Hydrolysis
  • In Vitro Techniques
  • Kinetics
  • Phosphatidylinositol 4,5-Diphosphate
  • Phosphatidylinositol Phosphates / biosynthesis*
  • Phosphatidylinositols / biosynthesis*
  • Phospholipids / metabolism
  • Thrombin / pharmacology*
  • Type C Phospholipases / metabolism*

Substances

  • Aminoquinolines
  • Phosphatidylinositol 4,5-Diphosphate
  • Phosphatidylinositol Phosphates
  • Phosphatidylinositols
  • Phospholipids
  • phosphatidylinositol 3,4-diphosphate
  • Type C Phospholipases
  • Thrombin
  • Quin2