Treatment of myelodysplastic syndromes with daily oral idarubicin. A phase I-II study

Cancer. 1993 Mar 15;71(6):1989-92. doi: 10.1002/1097-0142(19930315)71:6<1989::aid-cncr2820710611>3.0.co;2-t.

Abstract

Background: Idarubicin, a new anthracycline analogue, is available in an oral preparation, and responses have been observed using relatively aggressive therapy in patients with myelodysplastic syndromes (MDS). The authors studied whether a chronic low-dose schedule would be effective but less myelotoxic.

Methods: Forty-two patients with MDS received daily low-dose oral idarubicin in 5-week courses that included 3 weeks of treatment, followed by a 2-week rest period. Doses were escalated when possible after the second course, and each patient was to receive six courses.

Results: Only one partial response was observed. Although no patient had fatal bone marrow toxicity, only eight patients received the full six courses, primarily because of myelosuppression.

Conclusions: This schedule of oral idarubicin is relatively safe but produces fewer responses than are reported with the high-dose pulse regimens.

Publication types

  • Clinical Trial
  • Clinical Trial, Phase I
  • Clinical Trial, Phase II
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Administration, Oral
  • Drug Administration Schedule
  • Humans
  • Idarubicin / administration & dosage
  • Idarubicin / adverse effects
  • Idarubicin / therapeutic use*
  • Myelodysplastic Syndromes / drug therapy*

Substances

  • Idarubicin