Effects of the anti-gastric secretory drugs IT-066 and omeprazole mitogenic activities in the gastric juice of the rat

Scand J Gastroenterol. 1996 Feb;31(2):111-7. doi: 10.3109/00365529609031973.

Abstract

Background: Salivary epidermal growth factor (EGF) retains its biologic function in gastric juice and may play a physiologic role. Little is know, however, about the existence of mitogens other than EGF and the constitutional alterations of these factors in gastric juice by anti-secretagogues.

Methods: The mitogenic activity was evaluated by measuring [3H]-thymidine incorporation, and the EGF contribution was determined by using a specific anti-rat EGF antibody. An H2-receptor antagonist (IT-066) and a proton pump inhibitor (omeprazole) were used to determine whether these drugs alter the relative composition of active mitogens in gastric juice.

Results: Normal gastric juice significantly increased DNA synthesis. This activity was suppressed by antibody (87-88%). Both drugs increased EGF concentrations and activity dose-dependently IT-066 specifically increased total amount and activity of EGF. Approximately 50% of this activity was reduced by boiling or antibody.

Conclusion: The major mitogenic activity of normal rat gastric juice depends on EGF, and antisecretory drugs enhance the mitogenic activity by preserving and including intraluminal mitogens than EGF.

MeSH terms

  • Animals
  • Anti-Ulcer Agents / pharmacology*
  • Cell Line
  • DNA Replication / drug effects
  • Dose-Response Relationship, Drug
  • Epidermal Growth Factor / metabolism
  • Gastric Juice / drug effects*
  • Gastric Juice / metabolism
  • Growth Substances / metabolism*
  • Histamine H2 Antagonists / pharmacology*
  • Immunoenzyme Techniques
  • Omeprazole / pharmacology*
  • Piperidines / pharmacology*
  • Pyridines / pharmacology*
  • Rats
  • Rats, Sprague-Dawley

Substances

  • Anti-Ulcer Agents
  • Growth Substances
  • Histamine H2 Antagonists
  • Piperidines
  • Pyridines
  • IT 066
  • Epidermal Growth Factor
  • Omeprazole