alphaIIb beta 3-integrin mediated adhesion of human platelets to a fibrinogen matrix triggers phospholipase C activation and phosphatidylinositol 3',4'-biphosphate accumulation

FEBS Lett. 1996 Jul 8;389(3):253-6. doi: 10.1016/0014-5793(96)00595-9.

Abstract

This study focused on the variations in phosphoinositide metabolism depending upon alphaIIbbeta3-integrin/fibrinogen interaction without previous activation of platelet agonist receptors. We found that adhesion of resting human platelets to immobilized fibrinogen stimulates phosphatidic acid production and a concomitant decrease in phosphatidylinositol 4',5'-bisphosphate. These results, and the absence of a transphosphatidylation reaction, argue in favor of the activation of a phospholipase C. Moreover, we observed the accumulation of phosphatidylinositol 3',4'-bisphosphate in adherent platelets as a consequence of the activation of a phosphatidylinositol 3-kinase. This effect was inhibited by ADP scavengers. Our results demonstrate that in adherent platelets, whereas phosphatidylinositol 3-kinase activation is controlled by both alphaIIbbeta-integrin engagement and released ADP, phospholipase C stimulation is triggered only by alphaIIbbeta-integrin/fibrinogen interaction.

MeSH terms

  • Adenosine Diphosphate / metabolism
  • Blood Platelets / metabolism*
  • Cyclooxygenase Inhibitors / pharmacology
  • Enzyme Activation
  • Extracellular Matrix / metabolism
  • Fibrinogen / metabolism*
  • Humans
  • Phosphatidylinositol 3-Kinases
  • Phosphatidylinositol 4,5-Diphosphate
  • Phosphatidylinositol Phosphates / metabolism*
  • Phosphatidylinositols / metabolism
  • Phosphotransferases (Alcohol Group Acceptor) / metabolism
  • Platelet Adhesiveness*
  • Platelet Glycoprotein GPIIb-IIIa Complex / pharmacology*
  • Type C Phospholipases / metabolism*

Substances

  • Cyclooxygenase Inhibitors
  • Phosphatidylinositol 4,5-Diphosphate
  • Phosphatidylinositol Phosphates
  • Phosphatidylinositols
  • Platelet Glycoprotein GPIIb-IIIa Complex
  • phosphatidylinositol 3,4-diphosphate
  • Adenosine Diphosphate
  • Fibrinogen
  • Phosphatidylinositol 3-Kinases
  • Phosphotransferases (Alcohol Group Acceptor)
  • Type C Phospholipases