Transcriptional activation of the human epidermal growth factor receptor promoter by human p53

Mol Cell Biol. 1996 Nov;16(11):6009-19. doi: 10.1128/MCB.16.11.6009.

Abstract

The human epidermal growth factor receptor (EGFR) promoter is activated by both wild-type and tumor-derived mutant p53. In this communication, we demonstrate that EGFR promoter sequence requirements for transactivation by wild-type and mutant p53 are different. Transient-expression assays with EGFR promoter deletions identified a wild-type human p53 response element, 5'-AGCTAGACGTCCGGGCAGCCCCCGGCG -3', from positions --265 to --239. Electrophoretic mobility shift analysis and DNase I footprinting assays indicated that wild-type p53 binds sequence specifically to the response element. Using circularly permuted DNA fragments containing the p53-binding site, we show that wild-type p53 binding induces DNA bending at this site. We further show that the EGFR promoter is also activated by tumor-derived p53 mutants p53-143A, p53-175H, p53-248W, p53-273H, and p53-281G. However, the transactivation by mutant p53 does not require the wild-type p53-binding site. The minimal EGFR promoter from positions --104 to --20 which does not contain the wild-type p53-binding site is transactivated by the p53 mutants but not by the wild-type protein, showing a difference in the mechanism of transactivation by wild-type and mutant p53. Transactivation of the EGFR promoter by p53 may represent a novel mechanism of cell growth regulation.

Publication types

  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, Non-P.H.S.
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Amino Acid Sequence
  • Base Composition
  • Base Sequence
  • Binding Sites
  • Chloramphenicol O-Acetyltransferase / biosynthesis
  • ErbB Receptors / biosynthesis*
  • ErbB Receptors / genetics*
  • Humans
  • Molecular Sequence Data
  • Polymerase Chain Reaction
  • Promoter Regions, Genetic*
  • Recombinant Proteins / biosynthesis
  • Regulatory Sequences, Nucleic Acid
  • Restriction Mapping
  • Sequence Deletion
  • TATA Box
  • Transcriptional Activation*
  • Tumor Suppressor Protein p53 / metabolism*

Substances

  • Recombinant Proteins
  • Tumor Suppressor Protein p53
  • Chloramphenicol O-Acetyltransferase
  • ErbB Receptors